SCHEMBL9833995

SCHEMBL9833995

N#CC(C(=O)Nc1ccc(F)cc1)C(=O)c1nn(-c2ccc(Cl)cc2)c2c1COc1ccccc1-2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.41
CNR1 P21554 2/20 0.41
POLB P06746 2/20 0.41
PTGS1 P23219 1/20 0.40
PTGS2 P35354 1/20 0.40
IKBKB O14920 3/20 0.38
TP53 P04637 2/20 0.38
CYP1A2 P05177 1/20 0.37
HIF1A Q16665 1/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
CCNA2 P20248 2/20 0.36
CDK2 P24941 2/20 0.36
CCNA1 P78396 2/20 0.36
PIK3CD O00329 2/20 0.36
PIK3R2 O00459 2/20 0.36
PIK3CA P42336 2/20 0.36
PIK3CB P42338 2/20 0.36
PIK3CG P48736 2/20 0.36
PIK3R5 Q8WYR1 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9833080 0.96 MAPT (0.44) MAPTCNR1POLBPTGS1PTGS2
SCHEMBL9319611 0.93 MAPT (0.43) MAPTCNR1POLBPTGS1PTGS2
SCHEMBL9832762 0.93 MAPT (0.41) MAPTPOLBPTGS1PTGS2IKBKB
SCHEMBL9834264 0.92 MAPT (0.41) MAPTCNR1POLBIKBKBTP53
SCHEMBL9833393 0.92 ALDH1A1 (0.40) MAPTCNR1POLBIKBKBALDH1A1
SCHEMBL9831820 0.91 MAPT (0.43) MAPTPOLBPTGS1PTGS2IKBKB
SCHEMBL9832537 0.91 LMNA (0.42) MAPTCNR1POLBIKBKBTP53
SCHEMBL9316748 0.88 MAPT (0.44) MAPTPOLBPTGS1PTGS2TP53
SCHEMBL9834065 0.87 RIPK1 (0.39) MAPTPOLBPTGS1PTGS2TP53
SCHEMBL9831070 0.87 NR1H4 (0.41) MAPTPOLBCYP1A2HIF1AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0274443-B1 HETEROARYL 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.r.l. (IT) 1991-05-29 EP disclosed
US-4816467-A BACTERICIDES, VIRICIDES FARMITALIA CARLO ERBA S.R.L (IT) 1989-03-28 US disclosed
EP-0274443-A1 Heteroaryl 3-oxo-propanenitrile derivatives and process for their preparation FARMITALIA CARLO ERBA S.r.l. (IT) 1988-07-13 EP disclosed