SCHEMBL9834136

SCHEMBL9834136

CC(=O)Nc1ccc2c(c1)NC(=O)C2(C)C

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 1/20 0.51
SMN1; SMN2 Q16637 5/20 0.49
PDK2 Q15119 2/20 0.46
PDK4 Q16654 1/20 0.46
PGR P06401 1/20 0.45
MAPK14 Q16539 2/20 0.44
MEN1 O00255 4/20 0.43
KMT2A Q03164 4/20 0.43
MAPT P10636 3/20 0.43
MAOA P21397 2/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
ALDH1A1 P00352 2/20 0.43
KDM4A O75164 1/20 0.43
POLB P06746 1/20 0.43
THRB P10828 1/20 0.43
RECQL P46063 1/20 0.43
TP53 P04637 1/20 0.42
HSD17B10 Q99714 1/20 0.42
HTT P42858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10696147 0.88 NQO2 (0.61) NQO2SMN1; SMN2PDK2PDK4PGR
SCHEMBL9313195 0.88 MAPK14 (0.47) NQO2SMN1; SMN2PDK2PDK4PGR
SCHEMBL10586429 0.86 MAPK14 (0.49) NQO2PDK2PDK4PGRMAPK14
SCHEMBL9376571 0.86 CYP26A1 (0.52) NQO2SMN1; SMN2MAPK14MEN1KMT2A
SCHEMBL9377394 0.83 RAB9A (0.53) PGRMAPK14MEN1KMT2AMAPT
SCHEMBL9377389 0.83 HDAC1 (0.49) NQO2SMN1; SMN2PGRMAPK14MAPT
SCHEMBL9313814 0.82 MAOA (0.45) PDK2PDK4PGRMAPK14MEN1
SCHEMBL6620114 0.82 CA12 (0.49) NQO2SMN1; SMN2PDK2MEN1KMT2A
SCHEMBL31714594 0.82 ALDH1A1 (0.48) NQO2SMN1; SMN2PDK2MEN1KMT2A
SCHEMBL9312304 0.81 GSK3B (0.53) SMN1; SMN2PDK2PDK4PGRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0161632-B1 PYRROLO-BENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION, MEDICAMENTS CONTAINING THEM AND INTERMEDIATES Roche Diagnostics GmbH (DE) 1991-04-10 EP disclosed
US-4963686-A INTERMEDIATES FOR INOTROPIC AGENTS BOEHRINGER MANNHEIM GMBH (DE) 1990-10-16 US disclosed
EP-0161632-A2 Pyrrolo-benzimidazoles, process for their preparation, medicaments containing them and intermediates Roche Diagnostics GmbH (DE) 1985-11-21 EP disclosed