SCHEMBL9834776

SCHEMBL9834776

O=C(F)c1ccc(Cl)cc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 3/20 0.62
CES1 P23141 3/20 0.62
TSHR P16473 2/20 0.59
ALOX15 P16050 1/20 0.59
CA1 P00915 2/20 0.56
CA2 P00918 2/20 0.56
GSK3B P49841 2/20 0.52
MAPK1 P28482 2/20 0.52
SRD5A2 P31213 1/20 0.52
L3MBTL1 Q9Y468 2/20 0.50
LMNA P02545 2/20 0.50
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50
MAPT P10636 1/20 0.50
CYP3A4 P08684 1/20 0.46
ATM Q13315 1/20 0.46
PTGS2 P35354 1/20 0.45
ERCC5 P28715 1/20 0.45
FEN1 P39748 1/20 0.45
HPGD P15428 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL102601 0.85 TSHR (0.47) CES2CES1TSHRALOX15CA1
SCHEMBL11196376 0.83 ALDH1A1 (0.47) CES2CES1TSHRALOX15CA1
SCHEMBL3446105 0.77 SRD5A2 (0.58) CES2CES1TSHRALOX15CA1
SCHEMBL51827 0.77 SRD5A2 (0.80) CES2CES1TSHRALOX15CA1
SCHEMBL9065412 0.77 SRD5A2 (0.80) CES2CES1TSHRALOX15CA1
SCHEMBL10697158 0.77 SRD5A2 (0.80) CES2CES1TSHRALOX15CA1
SCHEMBL16798463 0.77 CES2 (0.52) CES2CES1TSHRALOX15CA1
SCHEMBL273857 0.77 CES2 (1.00) CES2CES1TSHRALOX15CA1
SCHEMBL22832292 0.77 SRD5A2 (0.55) MAPK1SRD5A2L3MBTL1LMNAALDH1A1
SCHEMBL12212918 0.77 BCL2L1 (0.50) CES2CES1TSHRGSK3BL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 63 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114181074-B Preparation method of p-chlorobenzoyl fluoride 大连奇凯医药科技有限公司 2024-03-15 CN claimed
CN-115717009-B Perovskite ink and preparation method and application thereof 江苏集萃有机光电技术研究所有限公司 2023-11-14 CN claimed
CN-115717009-A Perovskite ink and preparation method and application thereof 江苏集萃有机光电技术研究所有限公司 2023-02-28 CN claimed
CN-114181074-A Preparation method of p-chlorobenzoyl fluoride 大连奇凯医药科技有限公司 2022-03-15 CN claimed
EP-0253837-B1 CATALYTIC METHOD FOR PRODUCING FLUOROAROMATIC COMPOUNDS USING BRANCHED ALKYL PYRIDINIUM SALTS MALLINCKRODT SPECIALTY CHEMICALS COMPANY (US) 1991-10-09 EP claimed
EP-0253838-B1 CATALYTIC METHOD FOR PRODUCING FLUOROAROMATIC COMPOUNDS USING N-SEC-ALKYL PYRIDINIUM SALTS MALLINCKRODT SPECIALTY CHEMICALS COMPANY (US) 1991-08-21 EP claimed
EP-0252964-B1 CATALYTIC METHOD FOR PRODUCING FLUOROAROMATIC COMPOUNDS USING SUBSTITUTED PYRIDINIUM SALTS MALLINCKRODT SPECIALTY CHEMICALS COMPANY (US) 1991-08-21 EP claimed
US-4973771-A Phase transfer catalysts MALLINCKRODT, INC. (US) 1990-11-27 US claimed
US-4973772-A Catalytic method for producing fluoroarmatic compounds using substituted pyridinium salts MALLINCKRODT, INC. (US) 1990-11-27 US claimed
EP-0253836-B1 PREPARATION OF FLUOROAROMATIC COMPOUNDS IN DISPERSION OF POTASSIUM FLUORIDE Mallinckrodt, Inc. (a Delaware corporation) (US) 1990-10-03 EP claimed
EP-0253836-A4 PREPARATION OF FLUOROAROMATIC COMPOUNDS IN DISPERSION OF POTASSIUM FLUORIDE. MALLINCKRODT INC (US) 1988-04-27 EP claimed
EP-0253837-A4 CATALYTIC METHOD FOR PRODUCING FLUOROAROMATIC COMPOUNDS USING BRANCHED ALKYL PYRIDINIUM SALTS. MALLINCKRODT INC (US) 1988-04-26 EP claimed
EP-0253836-A1 PREPARATION OF FLUOROAROMATIC COMPOUNDS IN DISPERSION OF POTASSIUM FLUORIDE. MALLINCKRODT INC (US) 1988-01-27 EP claimed
EP-0253837-A1 CATALYTIC METHOD FOR PRODUCING FLUOROAROMATIC COMPOUNDS USING BRANCHED ALKYL PYRIDINIUM SALTS. MALLINCKRODT INC (US) 1988-01-27 EP claimed
EP-0252964-A1 CATALYTIC METHOD FOR PRODUCING FLUOROAROMATIC COMPOUNDS USING SUBSTITUTED PYRIDINIUM SALTS. MALLINCKRODT INC (US) 1988-01-20 EP claimed
WO-1987004148-A1 CATALYTIC METHOD FOR PRODUCING FLUOROAROMATIC COMPOUNDS USING BRANCHED ALKYL PYRIDINIUM SALTS MALLINCKRODT, INC. (US) 1987-07-16 WO claimed
WO-1987004151-A1 PREPARATION OF FLUOROAROMATIC COMPOUNDS IN DISPERSION OF POTASSIUM FLUORIDE MALLINCKRODT, INC. (US) 1987-07-16 WO claimed
WO-1987004149-A1 PHASE TRANSFER CATALYSTS MALLINCKRODT, INC. (US) 1987-07-16 WO claimed
WO-1987004150-A1 CATALYTIC METHOD FOR PRODUCING FLUOROAROMATIC COMPOUNDS USING SUBSTITUTED PYRIDINIUM SALTS MALLINCKRODT, INC. (US) 1987-07-16 WO claimed
EP-0069598-B1 PREPARATION OF AROMATIC KETONES RAYCHEM CORPORATION (a California corporation) (US) 1984-12-19 EP claimed