SCHEMBL9834932

SCHEMBL9834932

Cc1nc2cc3c(cc2[nH]1)NC(=S)C3(C)C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.40
KDM4E B2RXH2 5/20 0.40
POLB P06746 4/20 0.40
HPGD P15428 3/20 0.40
ALDH1A1 P00352 5/20 0.39
AURKA O14965 1/20 0.39
AURKB Q96GD4 1/20 0.39
CHRNB2 P17787 1/20 0.37
CHRNA4 P43681 1/20 0.37
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
HSP90AA1 P07900 1/20 0.36
ESR2 Q92731 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
PGR P06401 1/20 0.35
GAA P10253 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9834966 0.81 AURKA (0.56) MAPTKDM4EPOLBHPGDALDH1A1
SCHEMBL10669526 0.80 CHRNB2 (0.39) MAPTKDM4EPOLBHPGDALDH1A1
SCHEMBL10669533 0.80 CHRNB2 (0.39) MAPTKDM4EPOLBHPGDALDH1A1
SCHEMBL9833638 0.76 PDE4A (0.66) MAPTKDM4EPOLBHPGDALDH1A1
Water SCHEMBL10470921 0.76 PDE4A (0.65) MAPTKDM4EPOLBHPGDALDH1A1
SCHEMBL9831413 0.74 CBFB (0.57) MAPTKDM4EHPGDGAARAB9A
SCHEMBL9833271 0.73 MAPT (0.57) MAPTKDM4EPOLBHPGDALDH1A1
SCHEMBL14392380 0.71 MAPT (0.45) MAPTKDM4EPOLBHPGDALDH1A1
SCHEMBL13041691 0.71 ALDH1A1 (0.59) MAPTKDM4EPOLBHPGDALDH1A1
Hydrochloric Acid SCHEMBL10554384 0.71 AR (0.42) MAPTKDM4EPOLBHPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0214592-B1 PYRROLOBENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THESE PRODUCTS Roche Diagnostics GmbH (DE) 1991-08-14 EP disclosed
US-4730003-A Tricyclic compounds for treating heart and circulatory diseases BOEHRINGER MANNHEIM GMBH (DE) 1988-03-08 US disclosed
EP-0214592-A2 Pyrrolobenzimidazoles, process for their preparation and medicaments containing these products Roche Diagnostics GmbH (DE) 1987-03-18 EP disclosed