SCHEMBL9834985

SCHEMBL9834985

C=CC[C@@](Cc1c[nH]c2ccccc12)(NC(=O)OC(C)(C)C)C(=O)OC

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 3/20 0.48
CTSL P07711 2/20 0.47
CTSS P25774 1/20 0.47
CTSK P43235 1/20 0.47
MAPT P10636 5/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
TP53 P04637 1/20 0.45
SSTR3 P32745 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HDAC3 O15379 3/20 0.43
HDAC4 P56524 3/20 0.43
HDAC1 Q13547 3/20 0.43
HDAC7 Q8WUI4 3/20 0.43
HDAC2 Q92769 3/20 0.43
HDAC10 Q969S8 3/20 0.43
HDAC11 Q96DB2 3/20 0.43
HDAC8 Q9BY41 3/20 0.43
HDAC6 Q9UBN7 3/20 0.43
HDAC9 Q9UKV0 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9834979 1.00 TACR1 (0.48) TACR1CTSLCTSSCTSKMAPT
SCHEMBL9832740 0.83 CCKBR (0.47)
SCHEMBL9832751 0.83 CCKBR (0.47)
SCHEMBL8225007 0.80 MAPT (0.52) CTSLCTSSCTSKMAPTMEN1
SCHEMBL9270557 0.79 CTSL (0.55) TACR1CTSLCTSSCTSKMAPT
SCHEMBL3020291 0.76 CTSL (0.59) TACR1CTSLCTSSCTSKMAPT
SCHEMBL9016089 0.76 CTSL (0.59) TACR1CTSLCTSSCTSKMAPT
SCHEMBL3020294 0.76 CTSL (0.59) TACR1CTSLCTSSCTSKMAPT
SCHEMBL8651829 0.76 CTSL (0.58) TACR1CTSLCTSSCTSKMAPT
SCHEMBL2193454 0.76 CTSL (0.55) TACR1CTSLCTSSCTSKMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0442878-A4 DERIVATIVES OF TRYPTOPHAN AS CCK ANTAGONISTS 1991-10-23 EP disclosed
EP-0442878-A1 DERIVATIVES OF TRYPTOPHAN AS CCK ANTAGONISTS ABBOTT LABORATORIES (US) 1991-08-28 EP disclosed
WO-1989010355-A1 DERIVATIVES OF TRYPTOPHAN AS CCK ANTAGONISTS ABBOTT LABORATORIES (US) 1989-11-02 WO disclosed
EP-0336356-A2 Derivatives of tryptophan as CCK antagonists ABBOTT LABORATORIES (US) 1989-10-11 EP disclosed