SCHEMBL9835322

SCHEMBL9835322

CCC(=O)Nc1nc2cc3c(cc2[nH]1)NC(=O)C3(C)C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.45
PDE4B Q07343 1/20 0.45
PDE4C Q08493 1/20 0.45
PDE4D Q08499 1/20 0.45
PDE3B Q13370 1/20 0.45
PDE3A Q14432 1/20 0.45
AURKA O14965 3/20 0.44
AURKB Q96GD4 3/20 0.44
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
ALDH1A1 P00352 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
SPHK2 Q9NRA0 1/20 0.38
SPHK1 Q9NYA1 1/20 0.38
TUBB4A P04350 2/20 0.37
TUBB P07437 2/20 0.37
TUBA3C P0DPH7 2/20 0.37
TUBA1B P68363 2/20 0.37
TUBA4A P68366 2/20 0.37
TUBB4B P68371 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9833536 0.91 NPC1 (0.45) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9834452 0.86 AURKA (0.49) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9834995 0.80 PDE4A (0.55) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL2489471 0.78 PDE3B (0.48) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL10558334 0.77 RAB9A (0.58) NPC1RAB9ASMN1; SMN2TUBB4ATUBB
SCHEMBL9834410 0.76 PDE4A (0.46) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9835173 0.76 PDE3B (0.54) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9835346 0.76 PDE3B (0.51) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9833659 0.75 LMNA (0.46) PDE4APDE4BPDE4CPDE4DPDE3B
SCHEMBL9834966 0.74 AURKA (0.56) PDE4APDE4BPDE4CPDE4DPDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0214592-B1 PYRROLOBENZIMIDAZOLES, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THESE PRODUCTS Roche Diagnostics GmbH (DE) 1991-08-14 EP disclosed
US-4730003-A Tricyclic compounds for treating heart and circulatory diseases BOEHRINGER MANNHEIM GMBH (DE) 1988-03-08 US disclosed
EP-0214592-A2 Pyrrolobenzimidazoles, process for their preparation and medicaments containing these products Roche Diagnostics GmbH (DE) 1987-03-18 EP disclosed