SCHEMBL983559

SCHEMBL983559

O=C(NC1CCNCC1)c1c[nH]c2c(-c3ccccc3OCC3CC3)ncnc12

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PTK2 Q05397 6/20 0.39
HTR4 Q13639 1/20 0.38
MELK Q14680 2/20 0.37
ROCK2 O75116 1/20 0.37
AURKA O14965 2/20 0.36
RPS6KB1 P23443 2/20 0.36
PBK Q96KB5 1/20 0.36
SSTR1 P30872 1/20 0.36
SSTR4 P31391 1/20 0.36
PARP1 P09874 1/20 0.36
MRGPRX1 Q96LB2 1/20 0.35
KDM1A O60341 1/20 0.35
PIM1 P11309 1/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ethoxycarbonyl Group SCHEMBL28786267 0.92 PTK2 (0.36) PTK2HTR4MELKROCK2SSTR1
Tert-Butyl Formate SCHEMBL27802920 0.92 SSTR1 (0.36) PTK2HTR4MELKROCK2SSTR1
SCHEMBL984646 0.91 ACKR3 (0.41) PTK2HTR4KDM1AALDH1A1KMT2A
SCHEMBL984599 0.90 BTK (0.39) PBKMRGPRX1KDM1A
SCHEMBL982008 0.90 BTK (0.40) PTK2MRGPRX1KMT2A
Hydrochloric Acid SCHEMBL986113 0.90 ACKR3 (0.41) PTK2HTR4KDM1AALDH1A1KMT2A
SCHEMBL983264 0.90 BTK (0.40) PTK2MRGPRX1MEN1ALDH1A1KMT2A
SCHEMBL983586 0.90 BTK (0.35) MELKROCK2MRGPRX1MEN1ALDH1A1
Hydrochloric Acid SCHEMBL985798 0.89 ACKR3 (0.38) PTK2HTR4KDM1AALDH1A1KMT2A
SCHEMBL981511 0.88 KDM1A (0.42) PTK2HTR4PBKKDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8445501-B2 Substituted 7-carboxamido-pyrrolo[3,2-d]pyrimidines TAKEDA GMBH (DE) 2013-05-21 US disclosed
US-20110021479-A1 PYRROLOPYRIMIDINECARBOXAMIDES NYCOMED GMBH (DE) 2011-01-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110021479-A1 PYRROLOPYRIMIDINECARBOXAMIDES PDE5A, PDE3A, PDE2A PTK2 4247/4885HTR4 1818/4885MELK 4873/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.