SCHEMBL9835704

SCHEMBL9835704

Cc1ccc(S(=O)(=O)N(CCCCN2C(=O)c3ccccc3C2=O)CCCOS(C)(=O)=O)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 4/20 0.46
KEAP1 Q14145 1/20 0.45
NFE2L2 Q16236 1/20 0.45
ACHE P22303 7/20 0.45
BCHE P06276 2/20 0.44
NPSR1 Q6W5P4 3/20 0.44
ALDH1A1 P00352 3/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
LMNA P02545 2/20 0.44
TDP1 Q9NUW8 1/20 0.44
HPGD P15428 1/20 0.43
GAA P10253 2/20 0.42
MMP2 P08253 1/20 0.42
MMP9 P14780 1/20 0.42
NPC1 O15118 1/20 0.41
TSHR P16473 1/20 0.41
NR2F2 P24468 1/20 0.41
MAPK1 P28482 1/20 0.41
HTT P42858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9837228 0.84 KEAP1 (0.41) MAOBKEAP1NFE2L2NPSR1ALDH1A1
SCHEMBL10425135 0.83 MAOB (0.40) MAOBKEAP1NFE2L2ACHENPSR1
SCHEMBL21071153 0.81 MAPT (0.54) MAOBACHEMEN1KMT2ATDP1
SCHEMBL8269374 0.80 TDP1 (0.53) MAOBACHEMEN1KMT2ATDP1
SCHEMBL14764990 0.80 TDP1 (0.53) MAOBACHEMEN1KMT2ATDP1
SCHEMBL28598566 0.79 MAPT (0.59) MAOBNPSR1MEN1KMT2AHPGD
SCHEMBL9827695 0.77 MMP2 (0.43) MAOBKEAP1NFE2L2NPSR1ALDH1A1
SCHEMBL14121528 0.77 VDR (0.52) MAOBNPSR1ALDH1A1TDP1HPGD
SCHEMBL10770035 0.76 VDR (0.55) NPSR1ALDH1A1KMT2ALMNATDP1
SCHEMBL10425256 0.76 MMP2 (0.42) MAOBKEAP1NFE2L2NPSR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0215319-B1 GEM-DIHALO-1,8-DIAMINO-4-AZA-OCTANES MERRELL DOW PHARMACEUTICALS INC. (US) 1991-10-16 EP claimed
US-4914240-A PROTECTING DIHALO BUTANEDIOL, REACTING WITH POTASSIUM PHTHALIMINDE, DEPROTECTING; MULTISTEP MERRELL DOW PHARMACEUTICALS INC. (US) 1990-04-03 US claimed
EP-0215319-A2 Gem-dihalo-1,8-diamino-4-aza-octanes MERRELL DOW PHARMACEUTICALS INC. (US) 1987-03-25 EP claimed