SCHEMBL9836635

SCHEMBL9836635

COC(=O)C1=Cc2cc(C(n3ccnc3)C(C)(C)C)sc2CC1

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 3/20 0.53
CYP26A1 O43174 15/20 0.38
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
CYP17A1 P05093 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9836789 0.89 TBXAS1 (0.67) TBXAS1CYP26A1CYP1A2CYP3A4CYP2D6
SCHEMBL9834671 0.82 TBXAS1 (0.80) TBXAS1CYP26A1CYP3A4CYP17A1KMT2A
SCHEMBL9835771 0.81 TBXAS1 (0.50) TBXAS1CYP17A1KMT2A
SCHEMBL9837432 0.77 TBXAS1 (0.36) TBXAS1
SCHEMBL9871091 0.73 TBXAS1 (0.36) TBXAS1
SCHEMBL9835676 0.73 TBXAS1 (0.76) TBXAS1
SCHEMBL9835519 0.71 TBXAS1 (0.77) TBXAS1
SCHEMBL9835661 0.69 TBXAS1 (0.46) TBXAS1CYP17A1KMT2A
SCHEMBL9836166 0.69 TBXAS1 (1.00) TBXAS1CYP26A1CYP3A4CYP17A1KMT2A
SCHEMBL9835558 0.68 TBXAS1 (0.63) TBXAS1CYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0240107-B1 THIANAPHTHENE DERIVATIVES, THEIR PRODUCTION AND USE Sankyo Company Limited (JP) 1991-08-21 EP disclosed
US-5021444-A Anticoagulants SANKYO COMPANY LIMITED (JP) 1991-06-04 US disclosed
US-4847272-A ANTICOAGULANTS SANKYO COMPANY LIMITED (JP) 1989-07-11 US disclosed
EP-0240107-A1 Thianaphthene derivatives, their production and use Sankyo Company Limited (JP) 1987-10-07 EP disclosed