SCHEMBL9837246

SCHEMBL9837246

NC1Oc2ccccc2Cc2cccnc21

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAOA P21397 6/20 0.41
MAOB P27338 6/20 0.41
HTR2A P28223 1/20 0.35
NISCH Q9Y2I1 2/20 0.34
HTR1A P08908 3/20 0.34
HTR1D P28221 3/20 0.34
LTA4H P09960 1/20 0.31
AOC2 O75106 5/20 0.31
DAO P14920 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9837005 0.81 MAOA (0.41) MAOAMAOBNISCHHTR1AHTR1D
SCHEMBL9835181 0.81 MAOA (0.41) MAOAMAOBHTR2ANISCHHTR1A
Hydrochloric Acid SCHEMBL9835668 0.79 MAOA (0.40) MAOAMAOBNISCHHTR1AHTR1D
SCHEMBL10706601 0.77 MAOA (0.38) MAOAMAOBNISCHHTR1AHTR1D
SCHEMBL9836246 0.69 MTNR1A (0.40) HTR1AHTR1D
SCHEMBL1917308 0.67 MAOB (0.48) MAOAMAOBHTR2ANISCHHTR1A
SCHEMBL1648508 0.67 MAOA (0.59) MAOAMAOB
SCHEMBL31151882 0.67 MAOA (0.59) MAOAMAOB
SCHEMBL28671200 0.67 MAOA (0.39) MAOAMAOBHTR2ANISCHAOC2
SCHEMBL6997509 0.65 HTR2A (0.66) HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0129879-B1 A [1] benzepino(3,4-b)pyridine derivative KYOWA HAKKO KOGYO CO., LTD. (JP) 1991-09-11 EP disclosed
US-4547496-A Antiulcer [1] benzepino[3,4-b]pyridine and compositions KYOWA HAKKO KOGYO CO., LTD. (JP) 1985-10-15 US disclosed
EP-0129879-A2 A [1] benzepino(3,4-b)pyridine derivative KYOWA HAKKO KOGYO CO., LTD. (JP) 1985-01-02 EP disclosed