SCHEMBL9837349

SCHEMBL9837349

Cn1cc(C(N)=O)c(=O)c2sc(-c3ccccc3)cc21

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 6/20 0.49
JAK2 O60674 3/20 0.45
JAK3 P52333 1/20 0.45
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
BTK Q06187 1/20 0.43
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40
HPGD P15428 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9837257 0.90 ALDH1A1 (0.46) IKBKBKDM4EMEN1ALDH1A1GAA
SCHEMBL9836660 0.82 ALDH1A1 (0.55) CYP1A2CYP2C9KDM4EMEN1ALDH1A1
SCHEMBL9836198 0.78 KDM4E (0.39) KDM4EALDH1A1GAA
SCHEMBL9834409 0.77 KDM4E (0.41) KDM4EKMT2A
SCHEMBL10737753 0.76 NPC1 (0.41) KDM4EALDH1A1GAAHPGDKMT2A
SCHEMBL6050600 0.71 KDM4E (0.43) KDM4EMEN1ALDH1A1GAAKMT2A
SCHEMBL10341064 0.70 KDM4E (0.71) KDM4EMEN1ALDH1A1KMT2A
SCHEMBL30542063 0.70 KDM4E (0.71) KDM4EMEN1ALDH1A1KMT2A
Water SCHEMBL9837052 0.70 KDM4E (0.42) KDM4EMEN1ALDH1A1GAAKMT2A
Hydrochloric Acid SCHEMBL29812500 0.69 KDM4E (0.41) IKBKBKDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0269295-B1 THERAPEUTIC AGENTS The Boots Company PLC (GB) 1991-06-26 EP disclosed
US-4877793-A CARDIOVASCULAR DISORDERS THE BOOTS COMPANY, PLC (GB) 1989-10-31 US disclosed
EP-0269295-A1 Therapeutic agents The Boots Company PLC (GB) 1988-06-01 EP disclosed