SCHEMBL9837728

SCHEMBL9837728

CC(C)c1ccc(C=CC(=O)O)cn1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P4HTM Q9NXG6 1/20 0.58
KDM4E B2RXH2 7/20 0.57
MAPK1 P28482 3/20 0.57
GCK P35557 1/20 0.47
ESR1 P03372 2/20 0.46
HCAR2 Q8TDS4 2/20 0.46
CA12 O43570 2/20 0.46
AKR1B10 O60218 2/20 0.46
CA1 P00915 2/20 0.46
CA2 P00918 2/20 0.46
CA3 P07451 2/20 0.46
AKR1B1 P15121 2/20 0.46
CA4 P22748 2/20 0.46
CA6 P23280 2/20 0.46
DPP4 P27487 2/20 0.46
CA5A P35218 2/20 0.46
CA7 P43166 2/20 0.46
CA9 Q16790 2/20 0.46
CA14 Q9ULX7 2/20 0.46
CA5B Q9Y2D0 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5511343 1.00 P4HTM (0.58) P4HTMKDM4EMAPK1GCKESR1
SCHEMBL13881346 0.87 GLA (0.46) P4HTMKDM4EMAPK1GCKESR1
SCHEMBL12074871 0.81 PAM (0.50) P4HTMKDM4EMAPK1GCKESR1
SCHEMBL10140600 0.79 P4HTM (0.33) P4HTMKDM4EMAPK1ESR1ESR2
SCHEMBL5508613 0.77 KDM4E (0.53) P4HTMKDM4EMAPK1GCKESR1
SCHEMBL19116260 0.77 GRM5 (0.49) KDM4EMAPK1ALDH1A1SMN1; SMN2HPGD
SCHEMBL1124260 0.77 P4HTM (0.64) P4HTMKDM4EMAPK1GCKESR1
SCHEMBL1124258 0.77 P4HTM (0.64) P4HTMKDM4EMAPK1GCKESR1
SCHEMBL8731557 0.77 P4HTM (0.68) P4HTMKDM4EMAPK1ESR1HCAR2
SCHEMBL6853074 0.77 P4HTM (0.68) P4HTMKDM4EMAPK1ESR1HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0210782-B1 PYRIDINE COMPOUNDS, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME Dainippon Pharmaceutical Co., Ltd. (JP) 1991-04-17 EP disclosed
US-4778796-A ω-(3-pyridyl)alkenamide derivatives and anti-allergenic pharmaceutical compositions containing same DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1988-10-18 US disclosed
EP-0210782-A2 Pyridine compounds, process for the preparation thereof and pharmaceutical composition containing the same Dainippon Pharmaceutical Co., Ltd. (JP) 1987-02-04 EP disclosed