SCHEMBL9839481

SCHEMBL9839481

Clc1ccc(C2CC2Br)cc1Cl

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 12/20 0.47
SLC6A2 P23975 9/20 0.47
SLC6A4 P31645 9/20 0.44
CYP2D6 P10635 1/20 0.41
KCNH2 Q12809 1/20 0.41
TP53 P04637 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
TSHR P16473 1/20 0.40
MAPK1 P28482 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9839488 1.00 SLC6A3 (0.47) SLC6A3SLC6A2SLC6A4CYP2D6KCNH2
SCHEMBL7366491 0.83 SLC6A2 (0.45) SLC6A3SLC6A2SLC6A4CYP2D6KCNH2
SCHEMBL28202984 0.80 SLC6A3 (0.49) SLC6A3SLC6A2SLC6A4CYP2D6KCNH2
SCHEMBL7004268 0.78 KDM1A (0.48) SLC6A3SLC6A2CYP2D6KCNH2CYP1A2
SCHEMBL7004269 0.78 KDM1A (0.48) SLC6A3SLC6A2CYP2D6KCNH2CYP1A2
SCHEMBL8146309 0.78 KDM1A (0.48) SLC6A3SLC6A2CYP2D6KCNH2CYP1A2
SCHEMBL7095292 0.78 KDM1A (0.48) SLC6A3SLC6A2CYP2D6KCNH2CYP1A2
SCHEMBL731263 0.76 SLC6A3 (0.42) SLC6A3SLC6A2SLC6A4
Methyl Alcohol SCHEMBL9515247 0.75 SLC6A3 (0.45) SLC6A3SLC6A2SLC6A4
Methyl Alcohol SCHEMBL9515250 0.75 SLC6A3 (0.45) SLC6A3SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0154528-B1 ALKENE, ALKYNE OR CYCLOALKYLENE DERIVATIVES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-12-11 EP disclosed
US-5032592-A Antiandrogens IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-07-16 US disclosed
US-4873329-A ANTIANDROGENS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-10-10 US disclosed
EP-0154528-A2 Alkene, alkyne or cycloalkylene derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1985-09-11 EP disclosed