SCHEMBL9840565

SCHEMBL9840565

CCc1noc(-c2cc3c(cn2)[nH]c2ccc(C(C)O)cc23)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIKFYVE Q9Y2I7 1/20 0.36
GABRA1 P14867 12/20 0.33
GABRG2 P18507 12/20 0.33
GABRB3 P28472 12/20 0.33
GABRA5 P31644 12/20 0.33
GABRA3 P34903 12/20 0.33
GABRA2 P47869 12/20 0.33
GABRA6 Q16445 9/20 0.33
GABRA4 P48169 8/20 0.33
GABRP O00591 7/20 0.33
GABRD O14764 7/20 0.33
GABRB1 P18505 7/20 0.33
GABRB2 P47870 7/20 0.33
GABRE P78334 7/20 0.33
GABRG1 Q8N1C3 7/20 0.33
GABRG3 Q99928 7/20 0.33
GABRQ Q9UN88 7/20 0.33
PLAT P00750 1/20 0.32
IDO1 P14902 1/20 0.31
TP53 P04637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9839910 0.88 GABRA1 (0.34) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL9839940 0.85 GABRA1 (0.36) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL9840612 0.83 GABRA1 (0.39) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL7491336 0.82 GABRP (0.49) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL9839834 0.82 GABRA1 (0.37) PIKFYVEGABRA1GABRG2GABRB3GABRA5
SCHEMBL9839924 0.82 PIKFYVE (0.36) PIKFYVEGABRA1GABRG2GABRB3GABRA5
SCHEMBL7485906 0.81 OPRL1 (0.34) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL10374410 0.81 KMT2A (0.40) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL10376614 0.80 GABRA1 (0.36) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL10734560 0.78 S1PR1 (0.35) GABRA1GABRG2GABRB3GABRA5GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0222693-B1 3-OXADIAZOLYL AND 3-CARBOXYLIC-ACID BETA-CARBOLINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS MEDICAMENTS SCHERING AKTIENGESELLSCHAFT (DE) 1991-04-17 EP disclosed
US-4778800-A ANXIOLYTIC, ANTICONVULSANT SCHERING AKTIENGESELLSCHAFT (DE) 1988-10-18 US disclosed