SCHEMBL9840874

SCHEMBL9840874

CCCc1cnc(-c2ccc(OC(=O)C(C)CCC)cc2)nc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.46
THRB P10828 3/20 0.46
SMN1; SMN2 Q16637 5/20 0.46
RARB P10826 1/20 0.45
RAB9A P51151 7/20 0.40
NPC1 O15118 6/20 0.40
TP53 P04637 2/20 0.40
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
HDAC9 Q9UKV0 1/20 0.39
HDAC5 Q9UQL6 1/20 0.39
ACACB O00763 3/20 0.39
KMT2A Q03164 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9840511 0.93 RARB (0.52) MAPTTHRBSMN1; SMN2RARBRAB9A
SCHEMBL9840906 0.92 RARB (0.57) MAPTTHRBSMN1; SMN2RARBRAB9A
SCHEMBL9840863 0.91 RARB (0.59) MAPTTHRBSMN1; SMN2RARBRAB9A
SCHEMBL9840494 0.91 RARB (0.59) MAPTTHRBSMN1; SMN2RARBRAB9A
SCHEMBL10719851 0.91 RARB (0.56) MAPTTHRBSMN1; SMN2RARBRAB9A
SCHEMBL9839752 0.91 RARB (0.59) MAPTTHRBSMN1; SMN2RARBRAB9A
SCHEMBL9840675 0.91 RARB (0.59) MAPTTHRBSMN1; SMN2RARBRAB9A
SCHEMBL9840520 0.89 MAPT (0.50) MAPTTHRBSMN1; SMN2RARBRAB9A
SCHEMBL9840370 0.86 MAPT (0.46) MAPTTHRBSMN1; SMN2RARBRAB9A
SCHEMBL9237261 0.86 MAPT (0.47) MAPTTHRBSMN1; SMN2RARBRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0220297-B1 NITROGEN-CONTAINING HETEROCYCLES MERCK PATENT GmbH (DE) 1991-12-11 EP disclosed
EP-0220297-A1 NITROGEN-CONTAINING HETEROCYCLES. MERCK PATENT GMBH (DE) 1987-05-06 EP disclosed
WO-1986006373-A1 NITROGEN-CONTAINING HETEROCYCLES MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1986-11-06 WO disclosed