SCHEMBL9842293

SCHEMBL9842293

CC(C)CC(=O)C(C(=O)O)C1CNCCN1C(c1ccccc1)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 12/20 0.39
OPRM1 P35372 3/20 0.38
DPP4 P27487 1/20 0.37
DPP7 Q9UHL4 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
CCR5 P51681 1/20 0.36
CHRM2 P08172 3/20 0.35
CHRM4 P08173 3/20 0.35
CHRM5 P08912 3/20 0.35
CHRM1 P11229 3/20 0.35
CHRM3 P20309 3/20 0.35
OPRK1 P41145 2/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
OPRL1 P41146 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9842330 0.77 OPRD1 (0.42) OPRD1OPRM1DPP4DPP7MEN1
SCHEMBL3919530 0.76 MEN1 (0.50) OPRD1OPRM1MEN1KMT2AOPRK1
SCHEMBL9842200 0.73 OPRD1 (0.42) OPRD1OPRM1MEN1KMT2AOPRK1
SCHEMBL9842337 0.73 OPRD1 (0.39) OPRD1OPRM1DPP4DPP7MEN1
SCHEMBL4153276 0.70 MEN1 (0.53) OPRD1OPRM1MEN1KMT2ACHRM2
SCHEMBL4153281 0.70 MEN1 (0.53) OPRD1OPRM1MEN1KMT2ACHRM2
SCHEMBL9842206 0.70 OPRD1 (0.40) OPRD1OPRM1MEN1KMT2AOPRK1
SCHEMBL9842205 0.69 OPRD1 (0.43) OPRD1OPRM1MEN1KMT2AOPRK1
SCHEMBL9842287 0.69 OPRD1 (0.39) OPRD1OPRM1MEN1KMT2AOPRK1
SCHEMBL5633854 0.69 OPRD1 (0.50) OPRD1OPRM1MEN1KMT2ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0461264-A1 ETHYNYLPHENYL DERIVATIVE, PRODUCTION THEREOF, AND REMEDY FOR DISEASES OF CIRCULATORY ORGANS CONTAINING THE SAME AS ACTIVE INGREDIENT KAKEN PHARMACEUTICAL CO., LTD. (JP) 1991-12-18 EP disclosed