SCHEMBL9842872

SCHEMBL9842872

CC(C)(C)c1ccc(NC(=O)c2cnoc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.59
HDAC11 Q96DB2 1/20 0.59
HDAC8 Q9BY41 1/20 0.59
HDAC6 Q9UBN7 1/20 0.59
TRPV1 Q8NER1 5/20 0.57
NPC1 O15118 3/20 0.57
RAB9A P51151 3/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
NAMPT P43490 1/20 0.57
KDR P35968 1/20 0.54
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
KDM4E B2RXH2 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP2C9 P11712 1/20 0.53
HPGD P15428 1/20 0.53
CYP2C19 P33261 1/20 0.53
NR1H4 Q96RI1 1/20 0.52
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9843014 0.85 NPC1 (0.60) HDAC3HDAC8HDAC6TRPV1NPC1
SCHEMBL9842954 0.81 NQO2 (0.54) NPC1RAB9AMEN1KMT2AKDM4E
SCHEMBL11435148 0.81 TRPV1 (0.56) HDAC3HDAC8HDAC6TRPV1NPC1
SCHEMBL7303163 0.81 HDAC3 (0.86) HDAC3HDAC11HDAC8HDAC6TRPV1
SCHEMBL8597230 0.80 NPC1 (0.56) NPC1RAB9AMEN1KMT2A
SCHEMBL9081513 0.80 TRPV1 (0.50) TRPV1NPC1RAB9ANAMPTMEN1
SCHEMBL8808773 0.80 MAPK1 (0.57) NPC1RAB9ASMN1; SMN2NAMPTKDR
SCHEMBL8811207 0.80 TP53 (0.54) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL892704 0.80 HTT (0.54) HDAC8HDAC6NPC1RAB9ANAMPT
SCHEMBL9843089 0.79 RAB9A (0.64) NPC1RAB9ASMN1; SMN2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0440503-A1 4-Isoxazolecarboxamide derivatives SYNTEX (U.S.A.) INC. (US) 1991-08-07 EP claimed