SCHEMBL9842940

SCHEMBL9842940

O=C(Nc1ccc(-c2ccc(Cl)cc2)s1)c1cnoc1

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 16/20 0.53
ESR1 P03372 1/20 0.41
ESRRG P62508 1/20 0.41
IKBKB O14920 1/20 0.40
CYP1A2 P05177 1/20 0.39
MAPK1 P28482 1/20 0.39
APOBEC3A P31941 1/20 0.39
APOBEC3G Q9HC16 1/20 0.39
IL2 P60568 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9842883 0.89 CNR1 (0.52) CNR1CYP1A2MAPK1APOBEC3AAPOBEC3G
SCHEMBL9842919 0.88 CYP1A2 (0.42) CNR1ESR1ESRRGCYP1A2MAPK1
SCHEMBL9842938 0.84 IL2 (0.39) CNR1CYP1A2MAPK1APOBEC3AAPOBEC3G
SCHEMBL9842822 0.84 NPC1 (0.43) CYP1A2MAPK1APOBEC3AAPOBEC3GIL2
SCHEMBL9842957 0.84 CNR1 (0.45) CNR1CYP1A2MAPK1APOBEC3AAPOBEC3G
SCHEMBL9842960 0.82 KDR (0.42) CNR1CYP1A2MAPK1APOBEC3AAPOBEC3G
SCHEMBL9842892 0.82 HDAC6 (0.44) IL2
SCHEMBL9842925 0.81 CNR1 (0.39) CNR1CYP1A2MAPK1APOBEC3AAPOBEC3G
SCHEMBL9843027 0.81 CNR1 (0.52) CNR1ESR1ESRRGCYP1A2MAPK1
SCHEMBL9842863 0.80 CNR1 (0.36) CNR1IL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0440503-A1 4-Isoxazolecarboxamide derivatives SYNTEX (U.S.A.) INC. (US) 1991-08-07 EP disclosed