SCHEMBL9842892

SCHEMBL9842892

O=C(Nc1ccc(-c2ccc(OC(F)(F)F)cc2)s1)c1cnoc1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 1/20 0.44
ERCC5 P28715 1/20 0.44
FEN1 P39748 1/20 0.44
CHEK1 O14757 1/20 0.43
ABL1 P00519 9/20 0.43
SCN10A Q9Y5Y9 1/20 0.41
JAK2 O60674 1/20 0.40
JAK1 P23458 1/20 0.40
TYK2 P29597 1/20 0.40
JAK3 P52333 1/20 0.40
TRPV1 Q8NER1 3/20 0.39
IL2 P60568 2/20 0.39
OPRM1 P35372 1/20 0.39
KCNH2 Q12809 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9842993 0.85 IL2 (0.48) HDAC6TRPV1IL2
SCHEMBL9843028 0.85 CNR1 (0.51) HDAC6CHEK1
SCHEMBL9842960 0.85 KDR (0.42) IL2
SCHEMBL9842919 0.82 CYP1A2 (0.42) IL2
SCHEMBL9842940 0.82 CNR1 (0.53) IL2
SCHEMBL9842938 0.81 IL2 (0.39) IL2
SCHEMBL9842822 0.81 NPC1 (0.43) IL2
SCHEMBL9842888 0.80 TRPV1 (0.60) ABL1TRPV1OPRM1KCNH2
SCHEMBL9842991 0.80 CNR1 (0.54) HDAC6TRPV1IL2
SCHEMBL9843027 0.78 CNR1 (0.52) HDAC6IL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0440503-A1 4-Isoxazolecarboxamide derivatives SYNTEX (U.S.A.) INC. (US) 1991-08-07 EP disclosed