SCHEMBL9842991

SCHEMBL9842991

COc1cccc(-c2ccc(NC(=O)c3cnoc3)s2)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 2/20 0.54
PRKACA P17612 1/20 0.48
ROCK1 Q13464 1/20 0.48
HDAC6 Q9UBN7 1/20 0.46
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
IKBKB O14920 2/20 0.43
HSD17B2 P37059 2/20 0.43
PTPN1 P18031 1/20 0.43
HSD17B1 P14061 1/20 0.43
IL2 P60568 1/20 0.42
MAPT P10636 3/20 0.42
MAPK1 P28482 2/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
TP53 P04637 1/20 0.41
CYP1A2 P05177 1/20 0.41
APOBEC3A P31941 1/20 0.41
APOBEC3G Q9HC16 1/20 0.41
TRPV1 Q8NER1 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9843028 0.89 CNR1 (0.51) CNR1PRKACAROCK1HDAC6NPC1
SCHEMBL9843027 0.86 CNR1 (0.52) CNR1HDAC6NPC1RAB9AHSD17B2
SCHEMBL9842919 0.81 CYP1A2 (0.42) CNR1NPC1RAB9AHSD17B2PTPN1
SCHEMBL9842925 0.80 CNR1 (0.39) CNR1NPC1RAB9AIL2MAPT
SCHEMBL9842940 0.78 CNR1 (0.53) CNR1IKBKBIL2MAPK1CYP1A2
SCHEMBL9842993 0.78 IL2 (0.48) HDAC6NPC1RAB9AIL2MAPK1
SCHEMBL9842883 0.78 CNR1 (0.52) CNR1IL2MAPK1CYP1A2APOBEC3A
SCHEMBL9842960 0.77 KDR (0.42) CNR1NPC1RAB9AIL2MAPT
SCHEMBL9842938 0.76 IL2 (0.39) CNR1NPC1RAB9APTPN1IL2
SCHEMBL9842957 0.75 CNR1 (0.45) CNR1NPC1RAB9AIL2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0440503-A1 4-Isoxazolecarboxamide derivatives SYNTEX (U.S.A.) INC. (US) 1991-08-07 EP disclosed