SCHEMBL9842993

SCHEMBL9842993

O=C(Nc1ccc(-c2ccc(C(F)(F)F)cc2)s1)c1cnoc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IL2 P60568 2/20 0.48
MCHR1 Q99705 2/20 0.39
STAT3 P40763 2/20 0.39
STAT1 P42224 1/20 0.38
DEGS1 O15121 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
MAPK11 Q15759 1/20 0.38
MAPK14 Q16539 1/20 0.38
NPC1 O15118 2/20 0.38
PTGS1 P23219 1/20 0.38
KCNQ3 O43525 1/20 0.38
KCNQ2 O43526 1/20 0.38
KCNE1 P15382 1/20 0.38
KCNQ1 P51787 1/20 0.38
TRPV1 Q8NER1 1/20 0.37
RAB9A P51151 1/20 0.37
PTPN2 P17706 1/20 0.37
PTPN11 Q06124 1/20 0.37
CYP1A2 P05177 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9842822 0.88 NPC1 (0.43) IL2DEGS1NPC1RAB9ACYP1A2
SCHEMBL9842892 0.85 HDAC6 (0.44) IL2HDAC6TRPV1
SCHEMBL9842919 0.84 CYP1A2 (0.42) IL2NPC1RAB9APTPN11CYP1A2
SCHEMBL9842940 0.84 CNR1 (0.53) IL2CYP1A2MAPK1APOBEC3AAPOBEC3G
SCHEMBL9842938 0.84 IL2 (0.39) IL2NPC1RAB9APTPN2PTPN11
SCHEMBL9843028 0.81 CNR1 (0.51) DEGS1HDAC6NPC1RAB9A
SCHEMBL9842960 0.81 KDR (0.42) IL2NPC1RAB9ACYP1A2MAPK1
SCHEMBL9843027 0.81 CNR1 (0.52) IL2HDAC4HDAC6NPC1RAB9A
SCHEMBL9842925 0.79 CNR1 (0.39) IL2NPC1RAB9ACYP1A2MAPK1
SCHEMBL9843014 0.79 NPC1 (0.60) STAT3HDAC6NPC1PTGS1KCNQ3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0440503-A1 4-Isoxazolecarboxamide derivatives SYNTEX (U.S.A.) INC. (US) 1991-08-07 EP disclosed