SCHEMBL9844153

SCHEMBL9844153

NC(=O)C(C(N)=O)C(c1ccccc1)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.48
CYP2D6 P10635 2/20 0.46
SRC P12931 1/20 0.46
LMNA P02545 3/20 0.44
MAPK1 P28482 2/20 0.44
CYP1A2 P05177 1/20 0.44
PKM P14618 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
ALOX5 P09917 1/20 0.44
CTSD P07339 1/20 0.43
CES2 O00748 1/20 0.43
CES1 P23141 1/20 0.43
SLC6A3 Q01959 3/20 0.42
DRD3 P35462 2/20 0.42
ADORA3 P0DMS8 1/20 0.42
EDNRB P24530 1/20 0.42
MC4R P32245 1/20 0.42
CYP2C19 P33261 1/20 0.42
MC3R P41968 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1742565 0.82 SRC (0.59) CYP2D6SRCLMNAMAPK1CYP1A2
SCHEMBL9844391 0.80 CTRB1 (0.42) LMNACYP1A2ALOX5CTSDCYP2C19
SCHEMBL5834050 0.79 LMNA (0.48) EPHX1CYP2D6SRCLMNAMAPK1
SCHEMBL15577857 0.79 DPP4 (0.50) EPHX1CYP2D6SRCLMNAMAPK1
SCHEMBL3611836 0.79 DPP4 (0.50) EPHX1CYP2D6SRCLMNAMAPK1
SCHEMBL11022438 0.79 CYP2D6 (0.56) EPHX1CYP2D6SRCLMNAMAPK1
SCHEMBL341787 0.77 ALOX5 (0.50) EPHX1CYP2D6SRCLMNAMAPK1
SCHEMBL23052844 0.77 ALOX5 (0.55) EPHX1CYP2D6SRCLMNAMAPK1
Hydrochloric Acid SCHEMBL3618508 0.77 DPP4 (0.48) EPHX1CYP2D6SRCLMNAMAPK1
SCHEMBL1537326 0.77 EPHX1 (0.46) EPHX1CYP2D6SRCLMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0433662-A2 Acat inhibitors WARNER-LAMBERT COMPANY (US) 1991-06-26 EP claimed
CN-1051733-A Acyl-CoA: cholesteryl transferase inhibitor WARNER LAMBERT CO (US) 1991-05-29 CN disclosed