SCHEMBL9844786

SCHEMBL9844786

CN(Cc1cc2c(O)nc(N)nc2n1C)c1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 8/20 0.60
TYMS P04818 2/20 0.56
FOLR1 P15328 2/20 0.56
SLC46A1 Q96NT5 2/20 0.56
KDM4E B2RXH2 1/20 0.56
TLR4 O00206 1/20 0.56
MEN1 O00255 1/20 0.56
ALDH1A1 P00352 1/20 0.56
LMNA P02545 1/20 0.56
TP53 P04637 1/20 0.56
GLA P06280 1/20 0.56
POLB P06746 1/20 0.56
HMGB1 P09429 1/20 0.56
MAPT P10636 1/20 0.56
FOLR2 P14207 1/20 0.56
HPGD P15428 1/20 0.56
ALOX15 P16050 1/20 0.56
ALOX12 P18054 1/20 0.56
GART P22102 1/20 0.56
APEX1 P27695 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9844842 0.87 DHFR (0.61) DHFRTYMS
SCHEMBL9844785 0.85 DHFR (0.55) DHFRTYMSFOLR1SLC46A1FOLR2
SCHEMBL9844840 0.84 DHFR (0.56) DHFRTYMSFOLR1SLC46A1FOLR2
SCHEMBL6337570 0.83 DHFR (0.77) DHFRTYMSFOLR1SLC46A1KDM4E
SCHEMBL9844853 0.82 FOLR1 (0.62) DHFRTYMSFOLR1SLC46A1KDM4E
SCHEMBL9844756 0.79 DHFR (0.56) DHFRTYMSFOLR1SLC46A1FOLR2
SCHEMBL9221596 0.77 DHFR (0.55) DHFRTYMSFOLR1SLC46A1KDM4E
SCHEMBL9844739 0.77 DHFR (0.62) DHFRTYMSFOLR1SLC46A1KDM4E
SCHEMBL15056952 0.77 DHFR (0.90) DHFRTYMSFOLR1SLC46A1KDM4E
SCHEMBL6340352 0.77 DHFR (0.90) DHFRTYMSFOLR1SLC46A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP claimed
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP disclosed