SCHEMBL9844756

SCHEMBL9844756

CC(Cc1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc1)c1cc2c(O)nc(N)nc2n1C

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DHFR P00374 11/20 0.56
TYMS P04818 1/20 0.48
FOLR2 P14207 2/20 0.47
FOLR1 P15328 2/20 0.47
GART P22102 2/20 0.47
SLC46A1 Q96NT5 2/20 0.47
SLC19A1 P41440 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9844785 0.85 DHFR (0.55) DHFRTYMSFOLR2FOLR1GART
SCHEMBL9844840 0.83 DHFR (0.56) DHFRTYMSFOLR2FOLR1GART
SCHEMBL9844911 0.82 DHFR (0.56) DHFRTYMS
SCHEMBL9844841 0.82 DHFR (0.56) DHFRTYMSFOLR2FOLR1GART
SCHEMBL9844847 0.80 TP53 (0.40) DHFR
SCHEMBL9844786 0.79 DHFR (0.60) DHFRTYMSFOLR2FOLR1GART
SCHEMBL9564175 0.78 DHFR (0.53) DHFRTYMS
SCHEMBL9538587 0.78 DHFR (0.61) DHFRTYMSFOLR2FOLR1GART
SCHEMBL9844817 0.77 DHFR (0.61) DHFRTYMSFOLR2FOLR1GART
SCHEMBL9844820 0.77 DHFR (0.61) DHFRTYMSFOLR2FOLR1GART

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP disclosed