SCHEMBL9844801

SCHEMBL9844801

Nc1nc(O)c2cc(CCc3ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc3)oc2n1

nearest known ligand 0.60

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
DHFR P00374 13/20 0.60
TYMS P04818 4/20 0.54
GART P22102 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9844787 0.95 DHFR (0.61) DHFRTYMSGART
SCHEMBL9844911 0.84 DHFR (0.56) DHFRTYMS
SCHEMBL9844878 0.82 GART (0.72) DHFRTYMSGART
SCHEMBL9844849 0.81 GART (0.67) DHFRTYMSGART
SCHEMBL9535831 0.81 GART (0.72) DHFRTYMSGART
SCHEMBL10405409 0.80 DHFR (0.63) DHFRGART
SCHEMBL9844785 0.79 DHFR (0.55) DHFRTYMSGART
SCHEMBL9220727 0.79 DHFR (0.79) DHFRTYMSGART
SCHEMBL9339136 0.79 GART (0.68) DHFRTYMSGART
SCHEMBL9844791 0.79 GART (0.73) DHFRGART

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0438261-A2 Condensed heterocyclic glutamic acid derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-07-24 EP disclosed