SCHEMBL9845203

SCHEMBL9845203

C#Cc1cc(-c2cc3c(cc2C)SC(C)(C)CC3(C)C)ccc1CCCCC(=O)OCC

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 1/20 0.35
CYP4A11 Q02928 1/20 0.35
GSTP1 P09211 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
RARA P10276 1/20 0.31
RARB P10826 1/20 0.31
RARG P13631 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9845179 0.95 CYP4F2 (0.36) CYP4F2CYP4A11GSTP1CYP1A2CYP3A4
SCHEMBL9845166 0.94 ALDH1A1 (0.32) CYP4F2CYP4A11RARARARBRARG
SCHEMBL9845177 0.89 CYP4F2 (0.31) CYP4F2CYP4A11RARARARBRARG
SCHEMBL9845186 0.73 KDM4E (0.31) CYP4F2CYP4A11
SCHEMBL8864864 0.73 HPGD (0.33) CYP4F2CYP4A11RARARARBRARG
SCHEMBL9845198 0.72 ALDH1A1 (0.34) CYP4F2CYP4A11
SCHEMBL8866010 0.72 CYP4F2 (0.32) CYP4F2CYP4A11RARARARBRARG
SCHEMBL8865333 0.72 RARA (0.35) CYP4F2CYP4A11CYP3A4RARARARB
SCHEMBL8865174 0.71 CYP3A4 (0.36) CYP4F2CYP4A11CYP3A4RARARARB
SCHEMBL8865478 0.71 CYP4F2 (0.34) CYP4F2CYP4A11RARARARBRARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0419131-A2 Acetylenes disubstituted with a phenyl group and a 2-substituted chromanyl, thiochromanyl or 1,2,3,4-tetrahydroquinolinyl group having retinoid-like activity ALLERGAN, INC. (US) 1991-03-27 EP disclosed