SCHEMBL9845166

SCHEMBL9845166

C#Cc1cc(-c2cc3c(cc2C)SC(C)(C)CC3(C)C)ccc1CCC(=O)OCC

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
CYP4F2 P78329 1/20 0.32
CYP4A11 Q02928 1/20 0.32
RARA P10276 1/20 0.32
RARB P10826 1/20 0.32
RARG P13631 1/20 0.32
RXRA P19793 1/20 0.31
RXRB P28702 1/20 0.31
RXRG P48443 1/20 0.31
PTPN1 P18031 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9845203 0.94 CYP4F2 (0.35) CYP4F2CYP4A11RARARARBRARG
SCHEMBL9845177 0.89 CYP4F2 (0.31) ALDH1A1GAACYP4F2CYP4A11RARA
SCHEMBL9845179 0.89 CYP4F2 (0.36) CYP4F2CYP4A11RARARARBRARG
SCHEMBL9845198 0.78 ALDH1A1 (0.34) ALDH1A1GAACYP4F2CYP4A11PTPN1
SCHEMBL9845186 0.73 KDM4E (0.31) ALDH1A1GAACYP4F2CYP4A11
SCHEMBL9007048 0.72 RARA (0.37) ALDH1A1GAARARARARBRARG
SCHEMBL9282153 0.71 CYP4F2 (0.40) CYP4F2CYP4A11RARARARBRARG
SCHEMBL8875274 0.70 CYP3A4 (0.41) CYP4F2CYP4A11RARARARBRARG
SCHEMBL8561089 0.68 RARA (0.34) RARARARBRARG
SCHEMBL8864864 0.68 HPGD (0.33) CYP4F2CYP4A11RARARARBRARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0419131-A2 Acetylenes disubstituted with a phenyl group and a 2-substituted chromanyl, thiochromanyl or 1,2,3,4-tetrahydroquinolinyl group having retinoid-like activity ALLERGAN, INC. (US) 1991-03-27 EP disclosed