SCHEMBL9846101

SCHEMBL9846101

CCc1cc(CCc2nc3c(F)ccc(F)c3o2)c(=O)[nH]c1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.38
MEN1 O00255 2/20 0.38
HPGD P15428 2/20 0.38
KMT2A Q03164 2/20 0.38
GLA P06280 2/20 0.37
TSHR P16473 1/20 0.37
RAB9A P51151 2/20 0.36
NPC1 O15118 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C19 P33261 1/20 0.36
MCL1 Q07820 1/20 0.36
HSD17B10 Q99714 2/20 0.35
TNKS O95271 1/20 0.33
PARP1 P09874 1/20 0.33
TNKS2 Q9H2K2 1/20 0.33
HCAR2 Q8TDS4 2/20 0.32
KDM4E B2RXH2 2/20 0.30
MAPT P10636 2/20 0.30
TP53 P04637 1/20 0.30
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6366768 0.87 ALDH1A1 (0.35) ALDH1A1MEN1HPGDKMT2AGLA
SCHEMBL9680867 0.85 MEN1 (0.36) ALDH1A1MEN1HPGDKMT2AGLA
SCHEMBL9846133 0.84 PIK3CD (0.42) ALDH1A1MEN1HPGDKMT2AGLA
SCHEMBL9280614 0.84 PIK3CD (0.42) ALDH1A1MEN1HPGDKMT2AGLA
SCHEMBL9283877 0.83 ALDH1A1 (0.39) ALDH1A1MEN1HPGDKMT2AGLA
SCHEMBL9280809 0.81 ALDH1A1 (0.38) ALDH1A1MEN1HPGDKMT2AGLA
SCHEMBL9846239 0.81 MEN1 (0.32) ALDH1A1MEN1HPGDKMT2AGLA
SCHEMBL9278111 0.77 PIK3CD (0.44) ALDH1A1MEN1HPGDKMT2AGLA
SCHEMBL9281338 0.77 PIK3CD (0.44) ALDH1A1MEN1HPGDKMT2AGLA
SCHEMBL9846224 0.75 PARP1 (0.37) ALDH1A1MEN1HPGDKMT2AGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0462800-A2 Inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1991-12-27 EP claimed
EP-0462800-A2 Inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1991-12-27 EP disclosed