SCHEMBL9846230

SCHEMBL9846230

CCc1cc(NCc2cc3ccccc3nc2OC)c(=O)[nH]c1C

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.41
MAPT P10636 7/20 0.41
KDM4E B2RXH2 4/20 0.41
ALDH1A1 P00352 4/20 0.39
GAA P10253 3/20 0.39
HIF1A Q16665 1/20 0.39
APAF1 O14727 1/20 0.39
RECQL P46063 1/20 0.39
PDE10A Q9Y233 5/20 0.39
IDH1 O75874 2/20 0.37
ALOX12 P18054 1/20 0.36
PDE5A O76074 1/20 0.36
EGFR P00533 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
POLB P06746 1/20 0.34
HDAC3 O15379 2/20 0.34
HDAC1 Q13547 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9681349 0.86 MAPT (0.40) BTKMAPTKDM4EALDH1A1GAA
SCHEMBL9333881 0.83 MAPT (0.35) MAPTKDM4EALDH1A1GAAHIF1A
SCHEMBL9281981 0.82 MAPT (0.37) MAPTKDM4EALDH1A1GAAHIF1A
SCHEMBL9246249 0.77 MAPT (0.32) MAPTKDM4EGAAAPAF1RECQL
SCHEMBL9846089 0.77 NPSR1 (0.38) MAPTKDM4EALDH1A1GAAHIF1A
SCHEMBL9246243 0.77 PDE1A (0.32) MAPTKDM4EGAAAPAF1RECQL
SCHEMBL9846139 0.76 CYP2C9 (0.37) MAPTKDM4EALDH1A1GAAAPAF1
SCHEMBL10919184 0.75 ALDH1A1 (0.50) BTKMAPTKDM4EALDH1A1GAA
SCHEMBL9846192 0.74 HCAR2 (0.40) MAPTKDM4EAPAF1RECQLIDH1
SCHEMBL9432527 0.73 NPSR1 (0.47) MAPTKDM4EALDH1A1GAAALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0462800-A2 Inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1991-12-27 EP disclosed