SCHEMBL9846240

SCHEMBL9846240

CCc1cnc(OC)c(C#N)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.41
PIK3CA P42336 5/20 0.37
KCNH2 Q12809 1/20 0.37
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
KDM5A P29375 1/20 0.35
KDM4C Q9H3R0 1/20 0.35
AAK1 Q2M2I8 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
HPGD P15428 1/20 0.34
CYP2C19 P33261 1/20 0.34
LRRK2 Q5S007 1/20 0.34
PIK3CD O00329 5/20 0.34
PIK3CB P42338 2/20 0.34
PIK3CG P48736 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21705945 0.87 GAA (0.36) GAAPIK3CAKCNH2PDE4APDE4B
SCHEMBL17776991 0.86 KDM4E (0.40) GAAAAK1CYP1A2CYP3A4CYP2D6
SCHEMBL18358104 0.82 LMNA (0.44) KCNH2PDE4BPDE4CPDE4DAAK1
SCHEMBL21400936 0.77 CHRNB2 (0.38) GAAKCNH2KDM5AKDM4CCYP1A2
SCHEMBL7215762 0.77 L3MBTL1 (0.37) GAAKDM5AKDM4CCYP1A2CYP3A4
SCHEMBL15046199 0.77 GAA (0.44) GAAPIK3CAAAK1CYP1A2CYP3A4
SCHEMBL25117929 0.75 LMNA (0.42) GAAPIK3CAKCNH2CYP2C9HPGD
SCHEMBL21412856 0.75 GAA (0.40) GAAPIK3CA
SCHEMBL20670341 0.75 GAA (0.40) GAAPIK3CAAAK1HPGDPIK3CD
SCHEMBL18839637 0.75 KDM4E (0.49) GAAPIK3CAAAK1HPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0462800-A2 Inhibitors of HIV reverse transcriptase MERCK & CO. INC. (US) 1991-12-27 EP disclosed