SCHEMBL9846345

SCHEMBL9846345

N#CN=C(N)Nc1ccc(C=O)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.41
EGFR P00533 2/20 0.41
ALDH5A1 P51649 1/20 0.35
ABAT P80404 1/20 0.35
ALDH1A1 P00352 1/20 0.35
SIGMAR1 Q99720 4/20 0.34
GRIN2D O15399 3/20 0.34
GRIN3B O60391 3/20 0.34
GRIN1 Q05586 3/20 0.34
GRIN2A Q12879 3/20 0.34
GRIN2B Q13224 3/20 0.34
GRIN2C Q14957 3/20 0.34
GRIN3A Q8TCU5 3/20 0.34
ADRA2A P08913 3/20 0.34
ADRA2B P18089 2/20 0.34
ADRA2C P18825 2/20 0.34
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33
POLB P06746 1/20 0.33
PARP10 Q53GL7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9701789 0.79 PEPD (0.48) KDM4EALDH1A1SIGMAR1GRIN2DGRIN3B
SCHEMBL1983930 0.77 NPC1 (0.50) KDM4EALDH1A1SIGMAR1ADRA2AADRA2B
SCHEMBL11236640 0.77 GRIN2D (0.58) KDM4EALDH1A1SIGMAR1GRIN2DGRIN3B
SCHEMBL1983932 0.77 NPC1 (0.50) KDM4EALDH1A1SIGMAR1ADRA2AADRA2B
SCHEMBL10112792 0.77 SIGMAR1 (0.58) SIGMAR1GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL11232538 0.77 GRIN2D (0.55) KDM4EALDH1A1SIGMAR1GRIN2DGRIN3B
SCHEMBL15094415 0.77 GRIN2D (0.55) KDM4EALDH1A1SIGMAR1GRIN2DGRIN3B
SCHEMBL15366862 0.74 MDM2 (0.44) KDM4EALDH1A1ADRA2AADRA2BADRA2C
SCHEMBL160935 0.74 MDM2 (0.44) KDM4EALDH1A1ADRA2AADRA2BADRA2C
SCHEMBL11227305 0.73 CRHBP (0.51) ALDH1A1SIGMAR1POLBMAPTCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0456093-A2 Biguanide derivatives and biocidal compositions containing them H.B. FULLER LICENSING & FINANCING, INC. (US) 1991-11-13 EP disclosed