SCHEMBL9847736

SCHEMBL9847736

CCCn1c(CC(=O)O)nc2cc(F)ccc21

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 1/20 0.53
AGTR2 P50052 1/20 0.53
TBXA2R P21731 12/20 0.50
THRB P10828 1/20 0.47
RECQL P46063 1/20 0.47
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
HDAC1 Q13547 1/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
RXFP1 Q9HBX9 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5096807 0.81 AGTR1 (0.46) AGTR1AGTR2TBXA2RMEN1KMT2A
SCHEMBL5109530 0.81 AGTR1 (0.48) AGTR1AGTR2TBXA2RMEN1KMT2A
SCHEMBL1520801 0.81 KMT2A (0.64) RECQLMEN1KMT2AKDM4EALDH1A1
Bromide SCHEMBL5929370 0.80 AGTR1 (0.47) AGTR1AGTR2TBXA2RMEN1KMT2A
SCHEMBL14266729 0.78 AGTR1 (0.48) AGTR1AGTR2TBXA2RRECQLMEN1
SCHEMBL22965270 0.71 TBXA2R (0.50) AGTR1AGTR2TBXA2RKMT2AKDM4E
SCHEMBL7447330 0.70 AGTR1 (0.48) AGTR1AGTR2MEN1KMT2AKDM4E
SCHEMBL5107769 0.70 TBXA2R (0.48) TBXA2R
SCHEMBL12466547 0.70 ALDH1A1 (0.66) MEN1KMT2AKDM4EALDH1A1
SCHEMBL3065442 0.69 AGTR1 (0.39) AGTR1AGTR2TBXA2RMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0433648-A1 Substituted pyrimidobenzimidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 1991-06-26 EP disclosed