SCHEMBL9848138

SCHEMBL9848138

COc1ccc(C2=NCCc3cc(OCCN(C)C)ccc32)cc1OC

nearest known ligand 0.61

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.54
LMNA P02545 2/20 0.54
CA1 P00915 4/20 0.52
CA2 P00918 4/20 0.52
CA7 P43166 4/20 0.52
CA9 Q16790 4/20 0.52
CA14 Q9ULX7 4/20 0.52
MAPK10 P53779 7/20 0.51
KDM4E B2RXH2 1/20 0.51
LSS P48449 1/20 0.51
MAPK8 P45983 1/20 0.47
MAPK9 P45984 1/20 0.47
MAPK14 Q16539 1/20 0.47
ESR1 P03372 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9312666 0.82 MAPT (0.53) ALDH1A1LMNACA1CA2CA7
SCHEMBL9311736 0.78 MAPK10 (0.61) ALDH1A1LMNACA1CA2CA7
SCHEMBL28180887 0.77 ALDH1A1 (0.76) ALDH1A1LMNACA1CA2CA7
SCHEMBL31011321 0.77 ALDH1A1 (0.76) ALDH1A1LMNACA1CA2CA7
Hydrochloric Acid SCHEMBL9312979 0.77 MAPK10 (0.60) ALDH1A1LMNACA1CA2CA7
SCHEMBL9312347 0.77 MAPK10 (0.63) ALDH1A1LMNACA1CA2CA7
SCHEMBL5353435 0.75 MAPK10 (0.60) ALDH1A1LMNACA1CA2CA7
Hydrochloric Acid SCHEMBL9311868 0.74 MAPK10 (0.59) ALDH1A1LMNACA1CA2CA7
SCHEMBL17144585 0.70 CA1 (0.66) ALDH1A1LMNACA1CA2CA7
SCHEMBL983184 0.69 CA1 (0.66) ALDH1A1LMNACA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0422328-A2 Substituted isoquinolines and their use Euro-Celtique S.A. (LU) 1991-04-17 EP disclosed
US-4956371-A PLATELET ACTIVATING FACTOR EUROCELTIQUE, S.A. (LU) 1990-09-11 US disclosed