SCHEMBL9848649

SCHEMBL9848649

COc1ccc(CC(Cc2ccccc2)C(=O)N[C@H](C(=O)N[C@H](C(=O)N[C@@H](CC(N)=O)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](CC(C)C)C(=O)O)C(C)C)C(C)C)cc1

nearest known ligand 0.58

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 11/20 0.55
MMP1 P03956 1/20 0.52
MMP2 P08253 1/20 0.52
MMP3 P08254 1/20 0.52
MMP9 P14780 1/20 0.52
MME P08473 1/20 0.51
BACE2 Q9Y5Z0 1/20 0.50
CTSD P07339 1/20 0.49
ACE P12821 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9848658 0.87 BACE1 (0.53) BACE1MMEBACE2CTSD
SCHEMBL9848673 0.82 BACE1 (0.53) BACE1MMEBACE2CTSD
SCHEMBL9848616 0.81 BACE1 (0.57) BACE1BACE2CTSD
SCHEMBL29798307 0.81 BACE1 (0.67) BACE1BACE2CTSD
SCHEMBL9848640 0.80 BACE1 (0.55) BACE1BACE2CTSD
SCHEMBL9848655 0.80 BACE1 (0.55) BACE1BACE2CTSD
SCHEMBL9848653 0.80 BACE1 (0.54) BACE1MMEBACE2CTSD
SCHEMBL9848690 0.79 OPRD1 (0.62) BACE1BACE2CTSD
SCHEMBL9848628 0.79 BACE1 (0.59) BACE1BACE2CTSD
SCHEMBL9848664 0.79 OPRD1 (0.61) BACE1BACE2CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0438873-A1 Inhibitor of ribonucleotide reductase of herpes viruses MERCK & CO. INC. (US) 1991-07-31 EP disclosed