SCHEMBL9849208

SCHEMBL9849208

N#Cc1nccc2ccc(CCP(=O)(O)O)cc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2D O15399 2/20 0.39
GRIN3B O60391 2/20 0.39
GRIN1 Q05586 2/20 0.39
GRIN2A Q12879 2/20 0.39
GRIN2B Q13224 2/20 0.39
GRIN2C Q14957 2/20 0.39
GRIN3A Q8TCU5 2/20 0.39
PLAU P00749 1/20 0.36
FDPS P14324 2/20 0.35
TLR7 Q9NYK1 1/20 0.33
SLC22A12 Q96S37 2/20 0.33
EGLN2 Q96KS0 2/20 0.32
EGLN1 Q9GZT9 2/20 0.32
CYP1A2 P05177 3/20 0.32
CYP2D6 P10635 3/20 0.32
CYP2C9 P11712 2/20 0.32
CYP2C19 P33261 2/20 0.32
CYP3A4 P08684 1/20 0.32
HIF1A Q16665 1/20 0.32
CCNC P24863 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9849284 0.77 FDPS (0.36) PLAUFDPS
SCHEMBL9849459 0.76 PLAU (0.42) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL9849065 0.76 PLAU (0.34) PLAUSLC22A12
SCHEMBL9849066 0.75 PLAU (0.33) PLAUSLC22A12
SCHEMBL9849122 0.69 CYP19A1 (0.46) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL23088349 0.67 USP8 (0.44)
SCHEMBL29792782 0.67 USP8 (0.44)
SCHEMBL28518453 0.67 USP8 (0.44) EGLN2CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL30576360 0.66 KDM4E (0.36)
SCHEMBL15124651 0.66 KDM4E (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0421436-A2 Substituted carboxytetrahydroisoquinolines and derivatives thereof having pharmaceutical activity WARNER-LAMBERT COMPANY (US) 1991-04-10 EP disclosed