SCHEMBL9849532

SCHEMBL9849532

COc1cc(-c2nc(NCCCn3ccnc3)ccc2C#N)cc(OC)c1OC

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.54
GAA P10253 4/20 0.54
ALDH1A1 P00352 4/20 0.54
HPGD P15428 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
QPCT Q16769 8/20 0.48
POLB P06746 2/20 0.48
LMNA P02545 1/20 0.48
TSHR P16473 1/20 0.48
CASP1 P29466 1/20 0.48
CLK1 P49759 1/20 0.48
CASP7 P55210 1/20 0.48
HSD17B10 Q99714 1/20 0.48
FNTA P49354 2/20 0.46
FNTB P49356 2/20 0.46
PGGT1B P53609 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.44
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
SCN9A Q15858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9849422 0.79 QPCT (0.57) KDM4EGAAALDH1A1HPGDSMN1; SMN2
SCHEMBL3631942 0.78 QPCT (0.52) KDM4EGAAALDH1A1HPGDSMN1; SMN2
SCHEMBL9849540 0.78 ALDH1A1 (0.58) KDM4EGAAALDH1A1HPGDSMN1; SMN2
SCHEMBL3631599 0.77 QPCT (0.50) KDM4EGAAALDH1A1HPGDSMN1; SMN2
SCHEMBL9849543 0.77 ALDH1A1 (0.49) KDM4EGAAALDH1A1HPGDSMN1; SMN2
SCHEMBL3630133 0.77 QPCT (0.54) KDM4EGAAALDH1A1HPGDSMN1; SMN2
SCHEMBL9849531 0.69 ALDH1A1 (0.67) KDM4EGAAALDH1A1HPGDSMN1; SMN2
SCHEMBL9849298 0.67 ALDH1A1 (0.72) KDM4EGAAALDH1A1HPGDSMN1; SMN2
SCHEMBL9849546 0.67 ALDH1A1 (0.58) KDM4EGAAALDH1A1HPGDSMN1; SMN2
SCHEMBL8379438 0.67 QPCT (0.50) ALDH1A1QPCTPOLBL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0446604-A2 Pyridine and related aza heterocycle derivatives as cardiovascular agents AMERICAN CYANAMID COMPANY (US) 1991-09-18 EP disclosed