SCHEMBL9849543

SCHEMBL9849543

N#Cc1ccc(NCCCn2ccnc2)nc1-c1cccc(C(F)(F)F)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.49
KDM4E B2RXH2 5/20 0.49
LMNA P02545 3/20 0.49
POLB P06746 3/20 0.49
HPGD P15428 3/20 0.49
HSD17B10 Q99714 3/20 0.49
CASP1 P29466 2/20 0.49
CASP7 P55210 2/20 0.49
TSHR P16473 1/20 0.49
CLK1 P49759 1/20 0.49
GAA P10253 6/20 0.46
QPCT Q16769 3/20 0.43
TDP1 Q9NUW8 2/20 0.43
CTSK P43235 1/20 0.43
KCNH2 Q12809 1/20 0.43
MAPT P10636 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
SCN9A Q15858 1/20 0.42
NAMPT P43490 3/20 0.42
SOD1 P00441 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9849422 0.88 QPCT (0.57) ALDH1A1KDM4ELMNAPOLBHPGD
SCHEMBL9849628 0.84 KDM4E (0.56) ALDH1A1KDM4ELMNAPOLBHPGD
SCHEMBL9849532 0.77 KDM4E (0.54) ALDH1A1KDM4ELMNAPOLBHPGD
SCHEMBL3631542 0.77 KDM4E (0.49) ALDH1A1KDM4ELMNAPOLBHPGD
SCHEMBL3633387 0.77 GSK3A (0.53) ALDH1A1KDM4ELMNAHSD17B10GAA
SCHEMBL3632700 0.76 GSK3A (0.48) ALDH1A1KDM4EHPGDGAAQPCT
SCHEMBL9849540 0.75 ALDH1A1 (0.58) ALDH1A1KDM4ELMNAPOLBHPGD
SCHEMBL3632000 0.74 SMN1; SMN2 (0.54) ALDH1A1KDM4EHPGDGAAQPCT
SCHEMBL3631375 0.74 CTSK (0.48) ALDH1A1KDM4ELMNAHPGDGAA
SCHEMBL3633391 0.74 GSK3A (0.54) ALDH1A1KDM4EHSD17B10GAAQPCT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0446604-A2 Pyridine and related aza heterocycle derivatives as cardiovascular agents AMERICAN CYANAMID COMPANY (US) 1991-09-18 EP disclosed