SCHEMBL9849648

SCHEMBL9849648

COC(=O)c1cc(CCCCCCc2c(N)nc(N)nc2O)cs1

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
FOLR2 P14207 2/20 0.37
FOLR1 P15328 2/20 0.37
GART P22102 2/20 0.37
SLC19A1 P41440 1/20 0.37
CYP2D6 P10635 1/20 0.36
DHFR P00374 4/20 0.35
DAO P14920 1/20 0.33
SLC46A1 Q96NT5 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9850000 0.99 FOLR2 (0.37) FOLR2FOLR1GARTSLC19A1CYP2D6
SCHEMBL9850059 0.97 FOLR2 (0.39) FOLR2FOLR1GARTSLC19A1CYP2D6
SCHEMBL9849678 0.92 DAO (0.38) FOLR2FOLR1GARTSLC19A1CYP2D6
SCHEMBL9850021 0.89 DAO (0.45) FOLR2FOLR1GARTSLC19A1CYP2D6
SCHEMBL9849722 0.87 DAO (0.46) FOLR2FOLR1GARTSLC19A1CYP2D6
SCHEMBL9849630 0.85 DAO (0.46) FOLR2FOLR1GARTSLC19A1CYP2D6
SCHEMBL9849601 0.81 DHFR (0.31) FOLR2FOLR1GARTSLC19A1DHFR
SCHEMBL9849797 0.80 DAO (0.51) FOLR2FOLR1GARTSLC19A1CYP2D6
SCHEMBL9341073 0.79 CYP4A11 (0.53) CYP2D6DHFR
SCHEMBL9849766 0.79 HPGD (0.44) FOLR1CYP2D6DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0415510-A2 L-glutamic acid derivatives THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1991-03-06 EP disclosed
US-4920125-A L-glutamic acid derivatives THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1990-04-24 US disclosed