SCHEMBL9851422

SCHEMBL9851422

CCCc1nc2nc(Cl)ccc2[nH]1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MARS2 Q96GW9 4/20 0.41
SIRT2 Q8IXJ6 1/20 0.40
ADORA3 P0DMS8 2/20 0.39
ADORA2A P29274 2/20 0.39
ADORA1 P30542 2/20 0.39
KDM4E B2RXH2 1/20 0.39
PRMT5 O14744 2/20 0.38
NOS3 P29474 1/20 0.37
NOS1 P29475 1/20 0.37
NOS2 P35228 1/20 0.37
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10439327 0.90 PARP1 (0.40) MARS2PRMT5NOS3NOS1NOS2
SCHEMBL9318815 0.86 GAA (0.47) MARS2SIRT2ADORA3ADORA2AADORA1
SCHEMBL17513504 0.83 RAD52 (0.44) MARS2SIRT2KDM4EPRMT5NOS3
SCHEMBL9090094 0.83 ADORA1 (0.40) ADORA3ADORA2AADORA1KDM4ENOS3
SCHEMBL19378102 0.80 CACNA1H (0.40) MARS2SIRT2KDM4EPRMT5NOS3
SCHEMBL19408174 0.79 PRMT5 (0.40) MARS2SIRT2PRMT5NOS3NOS1
SCHEMBL9977950 0.79 TDP1 (0.49) MARS2SIRT2KDM4EPRMT5KMT2A
Hydrochloric Acid SCHEMBL19377908 0.77 PRMT5 (0.39) MARS2SIRT2KDM4EPRMT5NOS3
SCHEMBL9851491 0.77 PRMT5 (0.42) ADORA3ADORA2AADORA1KDM4EPRMT5
SCHEMBL9851421 0.77 NOS1 (0.60) SIRT2ADORA3ADORA2AADORA1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0434038-A1 Fused imidazole derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-06-26 EP disclosed