SCHEMBL9977950

SCHEMBL9977950

OCc1nc2nc(Cl)ccc2[nH]1

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.49
KDM4E B2RXH2 1/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
PRMT5 O14744 2/20 0.42
SIRT2 Q8IXJ6 1/20 0.38
MARS2 Q96GW9 5/20 0.37
NPSR1 Q6W5P4 1/20 0.37
RHEB Q15382 6/20 0.37
GRIN2B Q13224 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19408174 0.81 PRMT5 (0.40) TDP1PRMT5SIRT2MARS2GRIN2B
SCHEMBL9318815 0.81 GAA (0.47) PRMT5SIRT2MARS2
Hydrochloric Acid SCHEMBL19377908 0.80 PRMT5 (0.39) TDP1KDM4EPRMT5SIRT2MARS2
SCHEMBL17513504 0.79 RAD52 (0.44) TDP1KDM4EMEN1KMT2APRMT5
SCHEMBL9851422 0.79 MARS2 (0.41) KDM4EKMT2APRMT5SIRT2MARS2
SCHEMBL19378102 0.76 CACNA1H (0.40) TDP1KDM4EMEN1KMT2APRMT5
SCHEMBL10439327 0.76 PARP1 (0.40) KMT2APRMT5MARS2
SCHEMBL2299823 0.75 PRMT5 (0.49) KDM4EPRMT5SIRT2MARS2GRIN2B
SCHEMBL23725578 0.74 PRMT5 (0.44) PRMT5SIRT2MARS2GRIN2B
SCHEMBL6299123 0.71 ALDH1A1 (0.44) TDP1PRMT5SIRT2MARS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3131905-B1 SPIRO UREA COMPOUNDS AS RSV ANTIVIRAL COMPOUNDS JANSSEN SCIENCES IRELAND UC (IE) 2018-02-28 EP disclosed
EP-3131905-B1 SPIRO UREA COMPOUNDS AS RSV ANTIVIRAL COMPOUNDS JANSSEN SCIENCES IRELAND UC (IE) 2018-02-28 EP disclosed
US-9890178-B2 Azabenzimidazoles as respiratory syncytial virus antiviral agents JANSSEN SCIENCES IRELAND UC (IE) 2018-02-13 US disclosed
US-9890178-B2 Azabenzimidazoles as respiratory syncytial virus antiviral agents JANSSEN SCIENCES IRELAND UC (IE) 2018-02-13 US disclosed
US-9738652-B2 Spiro urea compounds as RSV antiviral compounds JANSSEN SCIENCES IRELAND UC (IE) 2017-08-22 US disclosed
US-9738652-B2 Spiro urea compounds as RSV antiviral compounds JANSSEN SCIENCES IRELAND UC (IE) 2017-08-22 US disclosed
US-9738652-B2 Spiro urea compounds as RSV antiviral compounds JANSSEN SCIENCES IRELAND UC (IE) 2017-08-22 US disclosed
EP-3131905-A1 SPIRO UREA COMPOUNDS AS RSV ANTIVIRAL COMPOUNDS Janssen Sciences Ireland UC (IE) 2017-02-22 EP disclosed
US-20170044172-A1 SPIRO UREA COMPOUNDS AS RSV ANTIVIRAL COMPOUNDS JANSSEN INFECTIOUS DISEASES BVBA (BE) 2017-02-16 US disclosed
US-20170044172-A1 SPIRO UREA COMPOUNDS AS RSV ANTIVIRAL COMPOUNDS JANSSEN INFECTIOUS DISEASES BVBA (BE) 2017-02-16 US disclosed
US-9321767-B2 Azabenzimidazoles as respiratory syncytial virus antiviral agents JANSSEN SCIENCES IRELAND UC (IE) 2016-04-26 US disclosed
EP-2651933-B1 AZABENZIMIDAZOLES AS RESPIRATORY SYNCYTIAL VIRUS ANTIVIRAL AGENTS JANSSEN SCIENCES IRELAND UC (IE) 2016-03-16 EP disclosed
WO-2015158653-A1 SPIRO UREA COMPOUNDS AS RSV ANTIVIRAL COMPOUNDS JANSSEN SCIENCES IRELAND UC (IE) 2015-10-22 WO disclosed
WO-2015158653-A1 SPIRO UREA COMPOUNDS AS RSV ANTIVIRAL COMPOUNDS JANSSEN SCIENCES IRELAND UC (IE) 2015-10-22 WO disclosed
US-20150073012-A1 AZABENZIMIDAZOLES AS RESPIRATORY SYNCYTIAL VIRUS ANTIVIRAL AGENTS JANSSEN SCIENCES IRELAND UC (IE) 2015-03-12 US disclosed
US-20150073012-A1 AZABENZIMIDAZOLES AS RESPIRATORY SYNCYTIAL VIRUS ANTIVIRAL AGENTS JANSSEN SCIENCES IRELAND UC (IE) 2015-03-12 US disclosed
US-8927720-B2 Azabenzimidazoles as respiratory syncytial virus antiviral agents JANSSEN R&D IRELAND (IE) 2015-01-06 US disclosed
US-8927720-B2 Azabenzimidazoles as respiratory syncytial virus antiviral agents JANSSEN R&D IRELAND (IE) 2015-01-06 US disclosed
US-20130261151-A1 AZABENZIMIDAZOLES AS RESPIRATORY SYNCYTIAL VIRUS ANTIVIRAL AGENTS JANSSEN R & D IRELAND (IE) 2013-10-03 US disclosed
WO-2012080449-A1 AZABENZIMIDAZOLES AS RESPIRATORY SYNCYTIAL VIRUS ANTIVIRAL AGENTS JANSSEN R&D IRELAND (IE) 2012-06-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170044172-A1 SPIRO UREA COMPOUNDS AS RSV ANTIVIRAL COMPOUNDS REN, ZC3HAV1, SAV1 TDP1 4556/4885KDM4E 2253/4885MEN1 4113/4885
US-20150073012-A1 AZABENZIMIDAZOLES AS RESPIRATORY SYNCYTIAL VIRUS ANTIVIRAL AGENTS ZC3HAV1, AZI2, ZC3HAV1L TDP1 3193/4885KDM4E 1258/4885MEN1 1913/4885
US-20130261151-A1 AZABENZIMIDAZOLES AS RESPIRATORY SYNCYTIAL VIRUS ANTIVIRAL AGENTS ZC3HAV1, AZI2, ZC3HAV1L TDP1 3193/4885KDM4E 1258/4885MEN1 1913/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.