SCHEMBL9852188

SCHEMBL9852188

C[C@@H](O)[C@H]1C(=O)N2C(C(=O)O)=C(SCc3ccccc3)[C@H](CCN(C)Cc3ccccc3)[C@H]12

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ELANE P08246 4/20 0.37
ESR1 P03372 1/20 0.35
PTGS1 P23219 1/20 0.35
PDE4A P27815 1/20 0.35
HPGD P15428 1/20 0.34
CACNA1C Q13936 1/20 0.34
ACKR3 P25106 1/20 0.33
LIPE Q05469 1/20 0.33
MAOB P27338 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9852139 0.85 ELANE (0.32) ELANELIPE
SCHEMBL9852332 0.82 LMNA (0.38) ELANEESR1PTGS1PDE4AKDM4E
SCHEMBL8865797 0.81 RECQL (0.36) ELANEESR1PTGS1PDE4AKDM4E
SCHEMBL9852265 0.81 RECQL (0.36) ELANEESR1PTGS1PDE4AKDM4E
SCHEMBL21081301 0.80 ESR1 (0.48) ELANEESR1PTGS1PDE4ACACNA1C
SCHEMBL9852153 0.79 ESR1 (0.34) ELANEESR1PTGS1PDE4AHPGD
SCHEMBL8865337 0.79 KDM4E (0.33) ELANEESR1PTGS1PDE4ACACNA1C
SCHEMBL9852063 0.78 LMNA (0.38) ELANEESR1PTGS1PDE4AKDM4E
SCHEMBL8864875 0.77 KDM4E (0.38) ELANEESR1PTGS1PDE4ACACNA1C
SCHEMBL9852179 0.76 LMNA (0.35) ELANEESR1PTGS1PDE4AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0433759-A1 4-Substituted alkyl carbapenem antibiotics Bristol-Myers Squibb Company (US) 1991-06-26 EP disclosed