SCHEMBL8865337

SCHEMBL8865337

C[C@@H](O)[C@H]1C(=O)N2C(C(=O)O)=C(SCc3ccncc3)[C@H](CCCCN(C)C)[C@H]12

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.33
ESR1 P03372 2/20 0.33
PTGS1 P23219 1/20 0.33
PDE4A P27815 1/20 0.33
CACNA1C Q13936 1/20 0.33
CHRM1 P11229 1/20 0.31
SLC6A4 P31645 1/20 0.31
KCNH2 Q12809 1/20 0.31
SLC29A1 Q99808 1/20 0.31
NPY2R P49146 1/20 0.31
ELANE P08246 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9852063 0.90 LMNA (0.38) KDM4ELMNAESR1PTGS1PDE4A
SCHEMBL9852079 0.89 KDM4E (0.36) KDM4ELMNAESR1PTGS1PDE4A
SCHEMBL9852089 0.88 KDM4E (0.36) KDM4ELMNAESR1PTGS1PDE4A
SCHEMBL8864875 0.86 KDM4E (0.38) KDM4ELMNAESR1PTGS1PDE4A
SCHEMBL9852072 0.84 CACNA1C (0.34) KDM4ELMNAESR1PTGS1PDE4A
SCHEMBL9852332 0.83 LMNA (0.38) KDM4ELMNAESR1PTGS1PDE4A
SCHEMBL9852407 0.82 CACNA1C (0.35) KDM4ELMNAESR1PTGS1PDE4A
SCHEMBL8865296 0.79 LMNA (0.35) KDM4ELMNAESR1PTGS1PDE4A
SCHEMBL9852143 0.79 CACNA1C (0.34) KDM4ELMNAESR1PTGS1PDE4A
SCHEMBL9852188 0.79 ELANE (0.37) KDM4EESR1PTGS1PDE4ACACNA1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5672701-A 4-substituted alkyl carbapenem antibiotics BRISTOL-MYERS SQUIBB COMPANY (US) 1997-09-30 US disclosed