SCHEMBL9852284

SCHEMBL9852284

CC(=O)Nc1nc(C)ns1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.53
L3MBTL1 Q9Y468 2/20 0.53
NPC1 O15118 3/20 0.51
RAB9A P51151 3/20 0.51
LMNA P02545 2/20 0.51
KMT2A Q03164 2/20 0.51
MEN1 O00255 1/20 0.51
POLB P06746 1/20 0.49
GRM1 Q13255 1/20 0.48
ADORA3 P0DMS8 1/20 0.47
MAPK1 P28482 1/20 0.46
MAPT P10636 3/20 0.46
ALDH1A1 P00352 2/20 0.46
HPGD P15428 2/20 0.46
HSD17B10 Q99714 2/20 0.46
ALOX15 P16050 1/20 0.46
DYRK1A Q13627 3/20 0.40
ADORA1 P30542 1/20 0.40
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9852290 0.85 SMN1; SMN2 (0.60) SMN1; SMN2L3MBTL1NPC1RAB9ALMNA
SCHEMBL3759738 0.85 GRM1 (0.49) SMN1; SMN2L3MBTL1NPC1RAB9ALMNA
SCHEMBL24491092 0.81 GRM1 (0.43) SMN1; SMN2L3MBTL1NPC1RAB9ALMNA
SCHEMBL24491053 0.79 SMN1; SMN2 (0.53) SMN1; SMN2L3MBTL1NPC1RAB9ALMNA
SCHEMBL24491070 0.79 SMN1; SMN2 (0.53) SMN1; SMN2L3MBTL1NPC1RAB9ALMNA
SCHEMBL24491025 0.79 RAB9A (0.56) SMN1; SMN2L3MBTL1NPC1RAB9ALMNA
SCHEMBL1855039 0.79 RAB9A (0.58) SMN1; SMN2NPC1RAB9ALMNAKMT2A
SCHEMBL16254891 0.75 SMN1; SMN2 (0.49) SMN1; SMN2L3MBTL1NPC1RAB9ALMNA
SCHEMBL9892988 0.75 SMN1; SMN2 (0.49) SMN1; SMN2L3MBTL1NPC1RAB9ALMNA
SCHEMBL9852268 0.75 NPC1 (0.53) SMN1; SMN2L3MBTL1NPC1RAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022117075-A1 AZACYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 广州费米子科技有限责任公司 2022-06-09 WO disclosed
EP-0455356-A1 Substituted 5-amino-1,2,4-thiadiazoles with pharmaceutical activity LILLY INDUSTRIES LIMITED (GB) 1991-11-06 EP disclosed