SCHEMBL9852492

SCHEMBL9852492

COc1ccc2c(c1)CCN(C(=O)CCc1cccs1)C2

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.53
ESR2 Q92731 1/20 0.53
RYR2 Q92736 1/20 0.51
ABHD6 Q9BV23 1/20 0.51
TAAR1 Q96RJ0 1/20 0.49
GAA P10253 2/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA7 P43166 1/20 0.47
CA9 Q16790 1/20 0.47
CA14 Q9ULX7 1/20 0.47
HCRTR1 O43613 1/20 0.47
HCRTR2 O43614 1/20 0.47
KMT2A Q03164 2/20 0.47
GFER P55789 1/20 0.47
CYP1A2 P05177 2/20 0.46
CYP2C19 P33261 2/20 0.46
TSHR P16473 1/20 0.46
MEN1 O00255 1/20 0.46
CYP2C9 P11712 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9852485 0.95 ESR1 (0.52) ESR1ESR2RYR2ABHD6TAAR1
SCHEMBL9852565 0.87 RAB9A (0.45) ESR1ESR2ABHD6TAAR1HCRTR1
SCHEMBL10398017 0.87 RAB9A (0.43) GAAHCRTR1HCRTR2CYP1A2CYP2C19
SCHEMBL9852572 0.84 ME2 (0.53) ESR1ESR2CA1CA2CA7
SCHEMBL28992968 0.79 KDM4E (0.57) TSHRALDH1A1
SCHEMBL10678740 0.78 ESR1 (0.59) ESR1ESR2RYR2ABHD6TAAR1
SCHEMBL10400059 0.77 ESR1 (0.64) ESR1ESR2RYR2ABHD6TAAR1
Hydrochloric Acid SCHEMBL9852489 0.76 KDM4E (0.54) TSHRALDH1A1
Hydrochloric Acid SCHEMBL9852486 0.75 KDM4E (0.53) TSHRALDH1A1
SCHEMBL3245803 0.74 ESR1 (0.64) ESR1ESR2RYR2ABHD6TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0422666-A2 6-Substituted-1,2,3,4-tetrahydroisoquinolines ABBOTT LABORATORIES (US) 1991-04-17 EP disclosed
US-4963563-A TREATING GLAUCOMA; INHIBITORS OF ALPHA-2-ADRENERGIC RECEPTORS ABBOTT LABORATORIES (US) 1990-10-16 US disclosed