SCHEMBL9852485

SCHEMBL9852485

COc1ccc2c(c1)CCN(C(=O)CCCc1cccs1)C2

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.52
ESR2 Q92731 1/20 0.52
RYR2 Q92736 1/20 0.50
TAAR1 Q96RJ0 1/20 0.48
ABHD6 Q9BV23 1/20 0.47
HRH3 Q9Y5N1 1/20 0.47
PKM P14618 2/20 0.47
ALDH1A1 P00352 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA7 P43166 1/20 0.47
CA9 Q16790 1/20 0.47
CA14 Q9ULX7 1/20 0.47
GAA P10253 1/20 0.47
HCRTR1 O43613 1/20 0.46
HCRTR2 O43614 1/20 0.46
LMNA P02545 1/20 0.46
KMT2A Q03164 1/20 0.46
NAMPT P43490 1/20 0.46
GFER P55789 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9852492 0.95 ESR1 (0.53) ESR1ESR2RYR2TAAR1ABHD6
SCHEMBL10398017 0.82 RAB9A (0.43) HRH3PKMALDH1A1GAAHCRTR1
SCHEMBL9852565 0.82 RAB9A (0.45) ESR1ESR2TAAR1ABHD6HRH3
Hydrochloric Acid SCHEMBL9852489 0.80 KDM4E (0.54) ALDH1A1TSHR
SCHEMBL9852572 0.79 ME2 (0.53) ESR1ESR2PKMALDH1A1CA1
SCHEMBL10678740 0.79 ESR1 (0.59) ESR1ESR2RYR2TAAR1ABHD6
Hydrochloric Acid SCHEMBL9852486 0.79 KDM4E (0.53) ALDH1A1TSHR
SCHEMBL28992968 0.78 KDM4E (0.57) ALDH1A1TSHR
SCHEMBL10400059 0.76 ESR1 (0.64) ESR1ESR2RYR2TAAR1ABHD6
SCHEMBL13504004 0.76 LMNA (0.61) PKMALDH1A1LMNAKMT2ANAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0422666-A2 6-Substituted-1,2,3,4-tetrahydroisoquinolines ABBOTT LABORATORIES (US) 1991-04-17 EP disclosed
US-4963563-A TREATING GLAUCOMA; INHIBITORS OF ALPHA-2-ADRENERGIC RECEPTORS ABBOTT LABORATORIES (US) 1990-10-16 US disclosed