SCHEMBL9853151

SCHEMBL9853151

C=Cc1sccc1C(=O)NO

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 7/20 0.42
HDAC6 Q9UBN7 5/20 0.42
HDAC8 Q9BY41 4/20 0.42
HDAC3 O15379 4/20 0.42
HDAC4 P56524 3/20 0.42
HDAC7 Q8WUI4 3/20 0.42
HDAC2 Q92769 3/20 0.42
HDAC10 Q969S8 3/20 0.42
HDAC11 Q96DB2 3/20 0.42
HDAC9 Q9UKV0 3/20 0.42
HDAC5 Q9UQL6 3/20 0.42
GAA P10253 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
KDM4E B2RXH2 2/20 0.41
MPO P05164 1/20 0.41
HIF1A Q16665 1/20 0.41
LIG1 P18858 1/20 0.38
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
MMP3 P08254 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9853209 0.79 MEN1 (0.43) GAASMN1; SMN2KDM4EALDH1A1MAPK1
SCHEMBL6048186 0.72 GAA (0.49) HDAC1HDAC6HDAC8HDAC3HDAC4
SCHEMBL3081395 0.68 HDAC1 (0.43) HDAC1HDAC6HDAC8HDAC3HDAC4
SCHEMBL12879068 0.66 PTPN1 (0.49) HDAC6GAASMN1; SMN2KDM4EMPO
SCHEMBL17255814 0.65 GAA (0.53) HDAC1HDAC6HDAC8HDAC3HDAC4
SCHEMBL21012218 0.65
SCHEMBL5176074 0.64 ALDH1A1 (0.52) HDAC1HDAC6HDAC8HDAC3HDAC4
SCHEMBL8637381 0.64 MCL1 (0.41) HDAC1HDAC6HDAC8HDAC3HDAC7
SCHEMBL10768728 0.63 HDAC1 (0.38) HDAC1HDAC6HDAC8HDAC3HDAC4
Ethane SCHEMBL28020377 0.63 GAA (0.50) HDAC1HDAC6HDAC8HDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0413293-A2 1-(Benzo[b]thienyl)-2-(thienyl) ethenes and related compounds, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1991-02-20 EP disclosed