SCHEMBL9853243

SCHEMBL9853243

c1ccc2c(c1)CNc1ccncc1O2

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.69
NPSR1 Q6W5P4 1/20 0.69
MAPT P10636 2/20 0.43
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
MAOA P21397 2/20 0.42
MAOB P27338 2/20 0.42
ALOX15 P16050 1/20 0.38
HSD17B10 Q99714 1/20 0.38
OXTR P30559 1/20 0.37
ALOX5 P09917 1/20 0.34
EGFR P00533 2/20 0.34
HTR5A P47898 2/20 0.33
IDO1 P14902 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
AURKA O14965 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
ACHE P22303 1/20 0.33
KDM4E B2RXH2 1/20 0.33
GABRP O00591 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL9853234 0.88 GAA (0.54) GAANPSR1MAPTKMT2AMEN1
Maleic Acid SCHEMBL9853230 0.88 GAA (0.54) GAANPSR1MAPTKMT2AMEN1
SCHEMBL1368071 0.82 GAA (1.00) GAANPSR1MAPTKMT2AMEN1
SCHEMBL14808600 0.75 MAOB (0.65) GAANPSR1KMT2AMEN1MAOA
Iodide SCHEMBL30281983 0.74 MAOB (0.63) GAANPSR1KMT2AMEN1MAOA
SCHEMBL8556344 0.72 NPSR1 (0.67) GAANPSR1MAPTKMT2AMEN1
SCHEMBL19810681 0.72 MAOA (0.48) GAANPSR1MAOAMAOBSMN1; SMN2
SCHEMBL8515984 0.72 MAOB (0.65) GAANPSR1KMT2AMEN1MAOA
SCHEMBL10593558 0.70 ALOX15 (0.66) GAANPSR1MAPTALOX15HSD17B10
SCHEMBL30704654 0.70 CA12 (0.46) GAANPSR1MAPTMAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4940704-A Pyrido[3,4-b][1,4]benzoxazepines HOECHST-ROUSSEL PHARMACEUTICAL INC. (US) 1990-07-10 US claimed
EP-0413300-A1 Pyrido [3,4-b][1,4] benzoxazepines, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1991-02-20 EP disclosed
US-4940704-A Pyrido[3,4-b][1,4]benzoxazepines HOECHST-ROUSSEL PHARMACEUTICAL INC. (US) 1990-07-10 US disclosed