SCHEMBL9854533

SCHEMBL9854533

CC(C(=O)C(F)(F)F)C(C)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.42
DPP7 Q9UHL4 1/20 0.42
HDAC4 P56524 3/20 0.41
HDAC6 Q9UBN7 3/20 0.41
HDAC3 O15379 2/20 0.41
HDAC1 Q13547 2/20 0.41
CES1 P23141 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
KEAP1 Q14145 1/20 0.39
NFE2L2 Q16236 1/20 0.39
CTRB1 P17538 2/20 0.39
CYP2D6 P10635 1/20 0.39
SRC P12931 1/20 0.39
ALOX5 P09917 1/20 0.38
LMNA P02545 2/20 0.38
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1033377 0.80 PTGS2 (0.47) HDAC4HDAC6HDAC3HDAC1CES1
SCHEMBL28842374 0.77 CYP2D6 (0.46) CES1KMT2ACYP2D6SRCALOX5
SCHEMBL585192 0.77 CYP2D6 (0.52) KEAP1NFE2L2CYP2D6SRCALOX5
SCHEMBL7787872 0.77 CYP2D6 (0.52) KEAP1NFE2L2CYP2D6SRCALOX5
SCHEMBL22351001 0.75 SRC (0.56) HDAC4HDAC6HDAC3HDAC1CES1
SCHEMBL15342224 0.75 CYP3A4 (0.49) DPP4CES1KMT2ACYP2D6SRC
SCHEMBL4568744 0.75 CYP3A4 (0.49) DPP4CES1KMT2ACYP2D6SRC
SCHEMBL6724975 0.75 CYP2D6 (0.44) CES1KMT2ACYP2D6SRCALOX5
SCHEMBL5692026 0.74 HDAC4 (0.49) DPP4DPP7HDAC4HDAC6HDAC3
SCHEMBL7475015 0.74 ALOX5 (0.55) CYP2D6SRCALOX5LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0253500-B1 ACYLANILIDE DERIVATIVES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1991-02-27 EP disclosed
US-4880839-A PROGESTATIONAL ACTIVITY IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-11-14 US disclosed
EP-0253500-A2 Acylanilide derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1988-01-20 EP disclosed