SCHEMBL9856069

SCHEMBL9856069

CSC(=O)c1cccc2c1NCCO2

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC11 Q96DB2 2/20 0.34
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC10 Q969S8 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
HDAC9 Q9UKV0 1/20 0.34
HDAC5 Q9UQL6 1/20 0.34
MTNR1A P48039 2/20 0.34
MTNR1B P49286 1/20 0.34
ADRA2A P08913 2/20 0.34
ADRA2C P18825 2/20 0.34
ADRA1D P25100 2/20 0.34
ADRA1A P35348 2/20 0.34
ADRA1B P35368 2/20 0.34
ADRA2B P18089 1/20 0.34
CTNNB1 P35222 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29804911 0.81 ALOX5 (0.46) HDAC11MTNR1AMTNR1BALDH1A1SMN1; SMN2
SCHEMBL749535 0.81 ALOX5 (0.46) HDAC11MTNR1AMTNR1BALDH1A1SMN1; SMN2
SCHEMBL22607785 0.80 PARP1 (0.45) HDAC11ALDH1A1MAPTHSD17B10KEAP1
SCHEMBL30517094 0.79 ALOX5 (0.51) ADRA1DADRA1AADRA1BCTNNB1WNT3A
SCHEMBL984368 0.79 ALOX5 (0.51) ADRA1DADRA1AADRA1BCTNNB1WNT3A
SCHEMBL9119474 0.77 ALDH1A1 (0.44) GAAALDH1A1MAPTSMN1; SMN2
SCHEMBL7940212 0.76 TSHR (0.49) ADRA1DADRA1AADRA1BGAAALDH1A1
SCHEMBL15621991 0.74 POLB (0.49) HDAC8HDAC6CTNNB1WNT3AGAA
SCHEMBL27602562 0.74 PARP1 (0.39) ALDH1A1MAPT
SCHEMBL13347539 0.73 MAPT (0.38) ALDH1A1MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0266849-B1 PROCESS FOR INTRODUCING A THIOCARBOXYLIC ESTER GROUP AT THE ORTHO-POSITION OF PHENOLS OR PHENYLAMINES SHIONOGI SEIYAKU KABUSHIKI KAISHA trading under the name of SHIONOGI & CO. LTD. (JP) 1991-03-13 EP disclosed
US-4857645-A Process for introducing a thiocarboxylic ester group at the orthoposition of phenols or phenylamines SHIONOGI & CO., LTD. (JP) 1989-08-15 US disclosed
EP-0266849-A1 Process for introducing a thiocarboxylic ester group at the ortho-position of phenols or phenylamines SHIONOGI SEIYAKU KABUSHIKI KAISHA trading under the name of SHIONOGI & CO. LTD. (JP) 1988-05-11 EP disclosed