SCHEMBL9857622

SCHEMBL9857622

Cc1cc(-c2cc(-c3ccccc3)cc(C)c2C(=O)O)ccc1F

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AKR1C2 P52895 2/20 0.42
AKR1C1 Q04828 1/20 0.42
PTGS2 P35354 2/20 0.41
DHODH Q02127 6/20 0.41
PTGS1 P23219 2/20 0.40
SRC P12931 1/20 0.40
PTPN1 P18031 1/20 0.40
ACMSD Q8TDX5 1/20 0.39
MCL1 Q07820 1/20 0.39
ALDH1A1 P00352 1/20 0.39
HSD17B10 Q99714 1/20 0.39
AKR1C3 P42330 1/20 0.38
MPL P40238 1/20 0.38
CAMKK2 Q96RR4 1/20 0.38
KAT6A Q92794 1/20 0.38
DHFR P00374 1/20 0.38
ALKBH5 Q6P6C2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9857916 0.87 AKR1C2 (0.39) AKR1C2AKR1C1PTGS2DHODHPTGS1
SCHEMBL9857473 0.87 DHODH (0.48) DHODHPTGS1PTPN1DHFRALKBH5
SCHEMBL17459516 0.86 PTPN1 (0.51) DHODHPTGS1PTPN1ALDH1A1HSD17B10
SCHEMBL9776295 0.85 PTGS2 (0.43) AKR1C2PTGS2PTGS1AKR1C3MPL
SCHEMBL10729814 0.79 MCL1 (0.49) MCL1ALDH1A1HSD17B10
SCHEMBL2882724 0.79 KDM4E (0.47) AKR1C2AKR1C1DHODHPTGS1PTPN1
SCHEMBL17459505 0.78 GFER (0.54) DHODHMCL1ALDH1A1
SCHEMBL5762155 0.77 ACHE (0.48) PTGS2PTGS1SRCALDH1A1
SCHEMBL9857687 0.77 PTGS2 (0.41) AKR1C2AKR1C1PTGS2DHODHPTGS1
SCHEMBL9857802 0.77 PTGS2 (0.44) PTGS2PTGS1SRCKAT6A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5072023-A Reacting lactone with ester anion to form cyclohexenone ester; oxidizing or dehydrogenating the intermediate E. R. SQUIBB & SONS, INC. (US) 1991-12-10 US disclosed
EP-0442495-A1 Process for preparing highly substituted phenyls E.R. SQUIBB & SONS, INC. (US) 1991-08-21 EP disclosed